SCHEMBL4060179

SCHEMBL4060179

Cc1ccc(C#N)c([NH])c1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.42
CYP2A6 P11509 2/20 0.41
ALDH1A1 P00352 1/20 0.41
TSHR P16473 1/20 0.38
PKM P14618 1/20 0.37
CYP11B1 P15538 2/20 0.36
CYP11B2 P19099 2/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
FFAR1 O14842 1/20 0.36
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1003862 0.78 ALDH1A1 (0.46) ARCYP2A6ALDH1A1TSHRPKM
SCHEMBL306406 0.77 AR (0.42) ARCYP2A6ALDH1A1TSHRPKM
SCHEMBL30361887 0.76 TSHR (0.52) ARCYP2A6ALDH1A1TSHRPKM
SCHEMBL277588 0.76 TSHR (0.52) ARCYP2A6ALDH1A1TSHRPKM
SCHEMBL8237072 0.74 AR (0.42) ARCYP2A6ALDH1A1TSHRPKM
SCHEMBL23192730 0.73 AR (0.42) ARCYP2A6ALDH1A1TSHRPKM
SCHEMBL2614496 0.73 TRPA1 (0.52) ARCYP2A6ALDH1A1TSHRCYP11B1
SCHEMBL21872468 0.73 AR (0.42) ARCYP2A6ALDH1A1TSHRPKM
SCHEMBL2434593 0.73 AR (0.46) ARCYP2A6ALDH1A1TSHRPKM
SCHEMBL410587 0.73 TRPV4 (0.57) ARCYP2A6ALDH1A1CYP11B2MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547713-B2 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives GU LIANQUAN 2009-06-16 US claimed
US-20060111405-A1 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives GU LIANQUAN 2006-05-25 US claimed
US-7547713-B2 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives GU LIANQUAN 2009-06-16 US disclosed
US-20060111405-A1 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives GU LIANQUAN 2006-05-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060111405-A1 O-pyridinequinone derivatives, the composition containing the derivatives, the process for preparation of the derivatives and the use of the derivatives PTGS2, PTGES2, PTGES AR 2202/4885CYP2A6 50/4885ALDH1A1 483/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.