SCHEMBL4065084

SCHEMBL4065084

O=C(c1ccccc1)c1ccc2nc(CCl)[nH]c2c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 4/20 0.64
ALDH1A1 P00352 3/20 0.64
POLB P06746 2/20 0.64
HPGD P15428 2/20 0.64
RAB9A P51151 2/20 0.64
SMN1; SMN2 Q16637 2/20 0.64
FABP6 P51161 1/20 0.64
HTT P42858 2/20 0.58
ABCC4 O15439 1/20 0.58
USP2 O75604 1/20 0.58
LMNA P02545 1/20 0.58
CYP1A2 P05177 1/20 0.58
CYP2C9 P11712 1/20 0.58
KDR P35968 1/20 0.58
HIF1A Q16665 1/20 0.58
ESR1 P03372 1/20 0.56
NPSR1 Q6W5P4 1/20 0.55
CHEK2 O96017 1/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4065081 0.89 KDM4E (0.51) ABL1ALDH1A1POLBHPGDRAB9A
SCHEMBL11277575 0.87 NPSR1 (0.72) ABL1ALDH1A1POLBHPGDRAB9A
SCHEMBL16134552 0.78 ABL1 (0.69) ABL1ALDH1A1POLBHPGDRAB9A
SCHEMBL3499235 0.78 ABL1 (1.00) ABL1ALDH1A1POLBHPGDRAB9A
SCHEMBL12909208 0.78 ALDH1A1 (1.00) ABL1ALDH1A1POLBHPGDRAB9A
SCHEMBL14642947 0.78 ABL1 (0.69) ABL1ALDH1A1POLBHPGDRAB9A
SCHEMBL29575638 0.78 ABL1 (1.00) ABL1ALDH1A1POLBHPGDRAB9A
SCHEMBL24329791 0.78 ALDH1A1 (0.60) ABL1ALDH1A1SMN1; SMN2HTTABCC4
SCHEMBL30469417 0.78 ALDH1A1 (0.60) ABL1ALDH1A1SMN1; SMN2HTTABCC4
SCHEMBL2243148 0.77 CHEK2 (0.80) ABL1ALDH1A1POLBHPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301422-A2 Thiomethyl and sulfinylmethyl derivatives having gastric acid antisecretory activity, processes for the preparation thereof and pharmaceutical compositions containing them CHIESI FARMACEUTICI S.p.A. (IT) 1989-02-01 EP claimed
EP-1317445-B1 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS ANORMED INC (CA) 2009-03-11 EP disclosed
US-7396840-B2 Chemokine receptor binding heterocyclic compounds GENZYME CORPORATION (US) 2008-07-08 US disclosed
US-7084155-B2 Chemokine receptor binding heterocyclic compounds ANORMED (CA) 2006-08-01 US disclosed
US-20060128750-A1 Chemokine receptor binding heterocyclic compounds GENZYME CORPORATION 2006-06-15 US disclosed
US-6864265-B2 Chemokine receptor binding heterocyclic compounds ANORMED, INC. (CA) 2005-03-08 US disclosed
US-20040220207-A1 Chemokine receptor binding heterocyclic compounds GENZYME CORPORATION 2004-11-04 US disclosed
CN-1457339-A Chemokine receptor binding heterocyclic compounds ANORMED INC (CA) 2003-11-19 CN disclosed
EP-1317445-A2 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS ANORMED INC. (CA) 2003-06-11 EP disclosed
US-20030018046-A1 Chemokine receptor binding heterocyclic compounds GENZYME CORPORATION 2003-01-23 US disclosed
WO-2002022600-A2 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS ANORMED INC. (CA) 2002-03-21 WO disclosed
US-5066652-A ANTIULCER AGENTS CHIESI FARMACEUTICI S.P.A. (IT) 1991-11-19 US disclosed
EP-0301422-A2 Thiomethyl and sulfinylmethyl derivatives having gastric acid antisecretory activity, processes for the preparation thereof and pharmaceutical compositions containing them CHIESI FARMACEUTICI S.p.A. (IT) 1989-02-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040220207-A1 Chemokine receptor binding heterocyclic compounds CXCR3, ACKR3, CCR2 ABL1 2316/4885ALDH1A1 1755/4885POLB 2246/4885
US-20060128750-A1 Chemokine receptor binding heterocyclic compounds CXCR4, CCR5, CXCR3 ABL1 1553/4885ALDH1A1 2001/4885POLB 2113/4885
US-20030018046-A1 Chemokine receptor binding heterocyclic compounds CXCR3, ACKR3, CCR2 ABL1 2316/4885ALDH1A1 1755/4885POLB 2246/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.