SCHEMBL4065194

SCHEMBL4065194

Cc1cc(Cl)ccc1Oc1ccc(NC(=O)c2ccccc2C)c(N)n1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.58
KCNMA1 Q12791 2/20 0.53
PNLIP P16233 1/20 0.51
GRM4 Q14833 1/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
KDM4E B2RXH2 3/20 0.46
SCN9A Q15858 1/20 0.46
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 2/20 0.45
ALOX15 P16050 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
METAP2 P50579 1/20 0.43
MAPT P10636 3/20 0.43
LMNA P02545 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
POLB P06746 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4064583 0.93 ALDH1A1 (0.49) ALDH1A1KCNMA1PNLIPGRM4NPC1
SCHEMBL4061920 0.90 ALDH1A1 (0.60) ALDH1A1KCNMA1PNLIPGRM4NPC1
SCHEMBL4069795 0.88 ALDH1A1 (0.43) ALDH1A1KDM4ESCN9AMEN1KMT2A
SCHEMBL4072610 0.85 TYK2 (0.42) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL4067700 0.83 ALDH1A1 (0.50) ALDH1A1KCNMA1PNLIPGRM4NPC1
SCHEMBL4062244 0.80 PNLIP (0.60) ALDH1A1PNLIPGRM4NPC1RAB9A
SCHEMBL4070607 0.75 RAB9A (0.41) ALDH1A1NPC1RAB9AKDM4EMEN1
SCHEMBL4069792 0.75 GRM8 (0.53) ALDH1A1PNLIPGRM4NPC1RAB9A
SCHEMBL4061271 0.74 PNLIP (0.58) ALDH1A1KCNMA1PNLIPGRM4NPC1
SCHEMBL4068452 0.74 CYP3A4 (0.44) ALDH1A1KDM4ESCN9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1028945-B9 SUBSTITUTED PYRIDINE COMPOUNDS AS ANTI-INFLAMMATORY AGENTS AMGEN INC (US) 2009-02-18 EP disclosed
EP-1028945-B1 SUBSTITUTED PYRIDINE COMPOUNDS AS ANTI-INFLAMMATORY AGENTS AMGEN INC (US) 2007-07-11 EP disclosed