SCHEMBL4070055

SCHEMBL4070055

CC(C)(C)[Si](C)(C)OCCN1C(=O)C(C(N)=O)Cc2ccc(Cl)cc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AADAT Q8N5Z0 2/20 0.38
MAPT P10636 2/20 0.32
KDM4E B2RXH2 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MEN1 O00255 1/20 0.32
CFTR P13569 1/20 0.32
UBE2I P63279 1/20 0.32
KMT2A Q03164 1/20 0.32
HKDC1 Q2TB90 1/20 0.32
GOPC Q9HD26 1/20 0.32
SAE1 Q9UBE0 1/20 0.32
UBA2 Q9UBT2 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
DUT P33316 1/20 0.32
CACNA1S Q13698 1/20 0.32
HTR2A P28223 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4075298 0.88 SMN1; SMN2 (0.33) MEN1UBE2IKMT2AHKDC1SAE1
SCHEMBL4067680 0.86 PYGL (0.36) AADATMAPTMEN1KMT2ATSHR
SCHEMBL4067889 0.86 AADAT (0.49) AADATMEN1KMT2ATSHRDUT
SCHEMBL13878903 0.86 AADAT (0.49) AADATMEN1KMT2ATSHRDUT
SCHEMBL4072393 0.80 DUT (0.39) TSHRDUTCACNA1SHTR2ASLC6A4
SCHEMBL4063656 0.80 AADAT (0.47) AADATMAPTL3MBTL1HTR2AHTR2C
SCHEMBL4063329 0.78 DUT (0.33) MEN1KMT2AHSD17B10DUT
SCHEMBL4071623 0.73 AADAT (0.37) AADATDUTBACE1
SCHEMBL13878891 0.73 AADAT (0.37) AADATDUTBACE1
SCHEMBL13878908 0.72 PYGL (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090099176-A1 PYRROLOPYRIDINE-2-CARBOXYLIC ACID AMIDES PROSIDION LIMITED (GB) 2009-04-16 US disclosed
EP-1819332-B1 PYRROLOPYRIDINE-2-CARBOXYLIC ACID AMIDES PROSIDION LTD (GB) 2009-03-11 EP disclosed
EP-1819332-A2 PYRROLOPYRIDINE-2-CARBOXYLIC ACID AMIDES Prosidion Limited (GB) 2007-08-22 EP disclosed
WO-2006059164-A2 PYRROLOPYRIDINE-2-CARBOXYLIC ACID AMIDES PROSIDION LIMITED (GB) 2006-06-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090099176-A1 PYRROLOPYRIDINE-2-CARBOXYLIC ACID AMIDES PC, GOT2, PDK1 AADAT 426/4885MAPT 3617/4885KDM4E 3425/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.