SCHEMBL4070973

SCHEMBL4070973

Cc1cc(-n2cc3c(n2)CCN(CC(=O)OC(C)(C)C)C3)ccn1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 9/20 0.44
KCNH2 Q12809 4/20 0.42
PDK2 Q15119 2/20 0.38
CDK9 P50750 4/20 0.36
CCNT1 O60563 3/20 0.36
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
WNT3A P56704 1/20 0.34
RXRA P19793 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13749198 0.87 SLC6A9 (0.45) SLC6A9KCNH2PDK2
Hydrochloric Acid SCHEMBL4067798 0.86 SLC6A9 (0.44) SLC6A9KCNH2PDK2
SCHEMBL4063883 0.84 MAPT (0.48) SLC6A9KCNH2PDK2MAPT
SCHEMBL13749100 0.81 SLC6A9 (0.42) SLC6A9KCNH2PDK2KDM4EMEN1
SCHEMBL13748459 0.81 SLC6A9 (0.44) SLC6A9KCNH2PDK2KDM4EMEN1
SCHEMBL13748801 0.79 SLC6A9 (0.41) SLC6A9KCNH2PDK2KDM4EMEN1
SCHEMBL13748458 0.79 SLC6A9 (0.44) SLC6A9KCNH2PDK2CDK9KDM4E
SCHEMBL13749073 0.79 SLC6A9 (0.39) SLC6A9KCNH2PDK2
SCHEMBL13748331 0.79 ALDH1A1 (0.47) SLC6A9KCNH2MEN1ALDH1A1MAPT
SCHEMBL13749141 0.79 SLC6A9 (0.43) SLC6A9KCNH2PDK2KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100120-A2 PYRIDINYL-SUBSTITUTED PIPERAZINYL OXOETHYL TETRAHYDROPYRAZOLOPYRIDINES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed
WO-2009100120-A2 PYRIDINYL-SUBSTITUTED PIPERAZINYL OXOETHYL TETRAHYDROPYRAZOLOPYRIDINES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed