SCHEMBL4078664

SCHEMBL4078664

O=C(Nc1n[nH]c2cc(C(=O)O)oc12)c1ccsc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.44
KCNK3 O14649 1/20 0.42
KCNK9 Q9NPC2 1/20 0.42
HDAC1 Q13547 1/20 0.39
LCK P06239 1/20 0.39
FYN P06241 1/20 0.39
DAO P14920 1/20 0.39
CDK2 P24941 2/20 0.38
CCNA2 P20248 1/20 0.38
CCNA1 P78396 1/20 0.38
GRM5 P41594 1/20 0.38
PARP1 P09874 1/20 0.38
GSK3B P49841 2/20 0.37
GSK3A P49840 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
CASP3 P42574 2/20 0.37
SENP8 Q96LD8 2/20 0.37
SENP7 Q9BQF6 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4083540 0.85 FGFR1 (0.50) FYNCDK2CCNA2CCNA1NPC1
SCHEMBL4088455 0.83 AURKA (0.47) HPGDKCNK3KCNK9GRM5NPC1
SCHEMBL4092896 0.82 HDAC6 (0.51) CDK2CCNA2CCNA1NPC1RAB9A
SCHEMBL3879252 0.82 GPR35 (0.45) KCNK3KCNK9CDK2CCNA2CCNA1
SCHEMBL4088586 0.81 KCNK3 (0.42) KCNK3KCNK9LCKPARP1GSK3B
SCHEMBL4081310 0.79 GPR35 (0.52) CDK2CCNA2CCNA1GSK3BNPC1
SCHEMBL4088257 0.79 AURKA (0.47) KCNK3FYNCDK2CCNA2CCNA1
SCHEMBL4088652 0.79 JAK2 (0.49) KCNK3KCNK9CDK2CCNA2CCNA1
SCHEMBL4088594 0.79 GPR35 (0.55) CDK2CCNA2CCNA1NPC1RAB9A
SCHEMBL4078387 0.79 MAPK1 (0.48) KCNK3KCNK9HDAC1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP disclosed