SCHEMBL4092896

SCHEMBL4092896

O=C(Nc1n[nH]c2cc(C(=O)O)oc12)c1ccc(Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 7/20 0.51
GPR35 Q9HC97 4/20 0.49
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
MAPT P10636 1/20 0.45
CLK2 P49760 3/20 0.45
DYRK1A Q13627 3/20 0.45
CDK2 P24941 2/20 0.45
STK17A Q9UEE5 2/20 0.45
CDC7 O00311 1/20 0.45
DAPK3 O43293 1/20 0.45
PAK4 O96013 1/20 0.45
FLT3 P36888 1/20 0.45
CSNK1A1 P48729 1/20 0.45
CDK7 P50613 1/20 0.45
CDK9 P50750 1/20 0.45
PRKX P51817 1/20 0.45
CDK5 Q00535 1/20 0.45
MELK Q14680 1/20 0.45
HIPK2 Q9H2X6 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4083540 0.89 FGFR1 (0.50) HDAC6GPR35NPC1RAB9ACLK2
SCHEMBL3879252 0.88 GPR35 (0.45) HDAC6GPR35NPC1RAB9AMAPT
SCHEMBL4088652 0.87 JAK2 (0.49) HDAC6GPR35NPC1RAB9ACLK2
SCHEMBL4081310 0.85 GPR35 (0.52) HDAC6GPR35NPC1RAB9ACLK2
SCHEMBL4088594 0.85 GPR35 (0.55) HDAC6GPR35NPC1RAB9ACDK2
SCHEMBL4081022 0.84 FLT3 (0.50) HDAC6GPR35NPC1RAB9AFLT3
SCHEMBL4078156 0.82 KDR (0.45) HDAC6NPC1RAB9AMAPTCDC7
SCHEMBL4082914 0.82 HRH3 (0.48) HDAC6RAB9AMAPTCLK2DYRK1A
SCHEMBL4092679 0.82 AURKA (0.49) HDAC6NPC1RAB9AMAPTCLK2
SCHEMBL4082126 0.82 HDAC6 (0.48) HDAC6GPR35NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP disclosed