SCHEMBL4088652

SCHEMBL4088652

O=C(Nc1n[nH]c2cc(C(=O)O)oc12)c1cccc(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.49
JAK1 P23458 1/20 0.49
NPC1 O15118 5/20 0.48
RAB9A P51151 3/20 0.48
CDK2 P24941 2/20 0.48
CDC7 O00311 2/20 0.48
DAPK3 O43293 1/20 0.48
PAK4 O96013 1/20 0.48
FLT3 P36888 1/20 0.48
CSNK1A1 P48729 1/20 0.48
CLK2 P49760 1/20 0.48
GSK3B P49841 1/20 0.48
CDK7 P50613 1/20 0.48
CDK9 P50750 1/20 0.48
PRKX P51817 1/20 0.48
CDK5 Q00535 1/20 0.48
DYRK1A Q13627 1/20 0.48
MELK Q14680 1/20 0.48
HIPK2 Q9H2X6 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4083540 0.88 FGFR1 (0.50) JAK2JAK1NPC1RAB9ACDK2
SCHEMBL4092896 0.87 HDAC6 (0.51) NPC1RAB9ACDK2CDC7DAPK3
SCHEMBL4088257 0.86 AURKA (0.47) JAK2NPC1RAB9ACDK2CDC7
SCHEMBL4091914 0.84 SMN1; SMN2 (0.51) JAK2NPC1RAB9ACDK2CDC7
SCHEMBL2913699 0.81 GPR35 (0.51) NPC1RAB9ACDK7GPR35MEN1
SCHEMBL3879252 0.80 GPR35 (0.45) NPC1RAB9ACDK2CDC7DAPK3
SCHEMBL4078664 0.79 HPGD (0.44) NPC1RAB9ACDK2GSK3BCDK7
SCHEMBL4088586 0.79 KCNK3 (0.42) RAB9AGSK3BHDAC6GPR35KCNK3
SCHEMBL4078387 0.79 MAPK1 (0.48) NPC1RAB9AHDAC6KCNK3KCNK9
SCHEMBL4081022 0.79 FLT3 (0.50) NPC1RAB9AFLT3HDAC6GPR35

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP disclosed