SCHEMBL4088586

SCHEMBL4088586

O=C(Nc1n[nH]c2cc(C(=O)O)oc12)c1ccoc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.42
KCNK9 Q9NPC2 1/20 0.42
PARP1 P09874 1/20 0.38
RAB9A P51151 1/20 0.38
TMIGD3 P0DMS9 1/20 0.37
ADORA1 P30542 1/20 0.37
GSK3B P49841 3/20 0.37
GSK3A P49840 1/20 0.37
ADORA3 P0DMS8 2/20 0.37
ADORA2A P29274 1/20 0.37
FGFR1 P11362 1/20 0.37
FGFR2 P21802 1/20 0.37
FGFR3 P22607 1/20 0.37
TBK1 Q9UHD2 1/20 0.36
LRRK2 Q5S007 4/20 0.36
HDAC6 Q9UBN7 1/20 0.36
LCK P06239 1/20 0.36
GPR35 Q9HC97 1/20 0.36
AURKA O14965 1/20 0.35
MAPK14 Q16539 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4083540 0.85 FGFR1 (0.50) RAB9AFGFR1FGFR2FGFR3HDAC6
SCHEMBL4078750 0.83 AURKA (0.45) KCNK3KCNK9PARP1ADORA3ADORA2A
SCHEMBL4092896 0.82 HDAC6 (0.51) RAB9AADORA3ADORA2AHDAC6GPR35
SCHEMBL3879252 0.82 GPR35 (0.45) KCNK3KCNK9RAB9AFGFR1FGFR2
SCHEMBL4078664 0.81 HPGD (0.44) KCNK3KCNK9PARP1RAB9AGSK3B
SCHEMBL4086303 0.80 MAPK1 (0.49) KCNK3KCNK9RAB9AADORA1ADORA3
SCHEMBL4088652 0.79 JAK2 (0.49) KCNK3KCNK9RAB9AADORA1GSK3B
SCHEMBL4081310 0.79 GPR35 (0.52) RAB9AGSK3BLRRK2HDAC6GPR35
SCHEMBL4088257 0.79 AURKA (0.47) KCNK3RAB9AFGFR1FGFR3AURKA
SCHEMBL4088594 0.79 GPR35 (0.55) RAB9AHDAC6GPR35AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP disclosed