SCHEMBL4093020

SCHEMBL4093020

COc1ccccc1C(=O)Nc1n[nH]c2cc(C(=O)NC(C)(C)c3ccccc3)oc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.44
MAP4K4 O95819 1/20 0.44
PIM1 P11309 1/20 0.44
CDK2 P24941 1/20 0.44
GSK3B P49841 1/20 0.44
HIPK2 Q9H2X6 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
ADORA3 P0DMS8 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
GPR35 Q9HC97 1/20 0.42
NPC1 O15118 6/20 0.41
AURKA O14965 1/20 0.41
RAB9A P51151 6/20 0.41
RXFP1 Q9HBX9 2/20 0.41
MAPT P10636 4/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
KCNK3 O14649 2/20 0.40
KCNK9 Q9NPC2 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL655164 0.87 AURKA (0.42) NPC1AURKARAB9ASMN1; SMN2
SCHEMBL4083477 0.87 AURKA (0.42) NPC1AURKARAB9AMAPTPKM
SCHEMBL4091966 0.86 GPR35 (0.54) CDC7MAP4K4PIM1CDK2GSK3B
SCHEMBL652230 0.86 RXFP1 (0.42) GPR35AURKARXFP1
SCHEMBL4088217 0.85 AURKA (0.51) CDK2AURKAROCK2ROCK1
SCHEMBL4082917 0.85 AURKA (0.48) CDK2ADORA3ADORA1GPR35NPC1
SCHEMBL653933 0.84 MEN1 (0.43) NPC1AURKARAB9ASMN1; SMN2
SCHEMBL4078482 0.84 HPGD (0.46) NPC1AURKARAB9AMAPTPKM
SCHEMBL4088617 0.84 CDK7 (0.46) CDC7MAP4K4CDK2HIPK2NPC1
SCHEMBL653327 0.84 AURKA (0.40) AURKARXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP disclosed