SCHEMBL4100878

SCHEMBL4100878

CCOc1ccc(CN=C(N)N)cc1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 5/20 0.58
NQO1 P15559 1/20 0.52
PARP10 Q53GL7 1/20 0.50
PRSS1 P07477 1/20 0.50
PRSS2 P07478 1/20 0.50
PRSS3 P35030 1/20 0.50
TSHR P16473 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
GRIN2D O15399 1/20 0.47
GRIN3B O60391 1/20 0.47
GRIN1 Q05586 1/20 0.47
GRIN2A Q12879 1/20 0.47
GRIN2B Q13224 1/20 0.47
GRIN2C Q14957 1/20 0.47
GRIN3A Q8TCU5 1/20 0.47
ALDH1A1 P00352 1/20 0.46
F11 P03951 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4093147 0.81 GRIN2B (0.65) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL1737052 0.79 GRIN1 (0.62) ADRA2AGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL9490727 0.78 NQO1 (0.64) ADRA2ANQO1PARP10PRSS1PRSS2
SCHEMBL4099965 0.73 ADRA2A (1.00) ADRA2ANQO1PARP10PRSS1PRSS2
1,4-Diethoxybenzene SCHEMBL28186701 0.72 NQO1 (1.00) ADRA2ANQO1PARP10PRSS1PRSS2
1,4-Diethoxybenzene SCHEMBL124015 0.72 NQO1 (1.00) ADRA2ANQO1PARP10PRSS1PRSS2
SCHEMBL2572011 0.72 PRSS1 (0.61) ADRA2ANQO1PARP10PRSS1PRSS2
SCHEMBL700166 0.72 PARP10 (0.61) NQO1PARP10TSHRTDP1ALDH1A1
SCHEMBL7635935 0.71 GRIN1 (0.54) ADRA2ATSHRTDP1GRIN2DGRIN3B
SCHEMBL4094076 0.71 GRIN2D (0.54) ADRA2AGRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090194124-A1 Hair Shaping Kit and Process Comprising at Least One Non-Hydroxide Imine MALLE GERARD 2009-08-06 US disclosed
US-20090139537-A1 HAIR RELAXING COMPOSITION COMPRISING AT LEAST ONE NON-HYDROXIDE IMINE L'OREAL S.A. 2009-06-04 US disclosed
US-20050136017-A1 Cosmetic containing an imine reactive with the cystines of keratin fibers via a beta-elimination reaction to produce dehydroalanine and lead to formation of lanthionine in a medium free of polyhydroxylated alkane; guanidine and/or amidine imines such as dimethylguanidine; noncaustic for use on hair, skin L'OREAL S.A. (FR) 2005-06-23 US disclosed
US-20050129645-A1 Hair shaping composition comprising at least one non-hydroxide imine L'OREAL 2005-06-16 US disclosed
EP-1532963-A1 Composition for straightening the hair comprising at least one imine not being an hydroxide L'OREAL (FR) 2005-05-25 EP disclosed
EP-1532960-A1 Hair styling composition containing a non-hydroxide imine L'OREAL (FR) 2005-05-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090139537-A1 HAIR RELAXING COMPOSITION COMPRISING AT LEAST ONE NON-HYDROXIDE IMINE KRT18, INMT, INHA ADRA2A 2119/4885NQO1 3017/4885PARP10 2162/4885
US-20090194124-A1 Hair Shaping Kit and Process Comprising at Least One Non-Hydroxide Imine KRT18, KIT, PRDM7 ADRA2A 4807/4885NQO1 1627/4885PARP10 3249/4885
US-20050129645-A1 Hair shaping composition comprising at least one non-hydroxide imine KRT18, INHA, H1-5 ADRA2A 4808/4885NQO1 1164/4885PARP10 3549/4885
US-20050136017-A1 Cosmetic containing an imine reactive with the cystines of keratin fibers via a beta-elimination reaction to produce dehydroalanine and lead to formation of lanthionine in a medium free of polyhydroxylated alkane; guanidine and/or amidine imines such as dimethylguanidine; noncaustic for use on hair, skin BHMT, KRT18, INMT ADRA2A 1818/4885NQO1 2408/4885PARP10 3537/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.