Pamoic Acid

Pamoic Acid

SCHEMBL41090

CN(C)CCCN1c2ccccc2CCc2ccccc21.O=C(O)c1cc2ccccc2c(Cc2c(O)c(C(=O)O)cc3ccccc23)c1O

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2DRD3DRD4GNRHRHRH1HTR2AHTR2CSLC6A2SLC6A4SSTR1SSTR2SSTR3SSTR5

The experimentally established mechanism targets of Pamoic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 known ✓ P31645 13/20 0.56
HRH1 known ✓ P35367 4/20 0.56
DRD2 known ✓ P14416 3/20 0.56
SLC6A2 known ✓ P23975 3/20 0.56
HTR2A known ✓ P28223 3/20 0.56
HTR2C known ✓ P28335 3/20 0.56
DRD3 known ✓ P35462 3/20 0.56
DRD4 known ✓ P21917 1/20 0.56
MAPT P10636 4/20 0.56
LMNA P02545 3/20 0.56
ADORA3 P0DMS8 3/20 0.56
CHRM1 P11229 3/20 0.56
ADRA2B P18089 3/20 0.56
ADRA2C P18825 3/20 0.56
CHRM3 P20309 3/20 0.56
ADRA1A P35348 3/20 0.56
OPRK1 P41145 3/20 0.56
SLC6A3 Q01959 3/20 0.56
KCNH2 Q12809 3/20 0.56
SLC22A1 O15245 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pamoic Acid SCHEMBL21834068 1.00 SLC6A4 (0.56) SLC6A4MAPTHRH1LMNAADORA3
Pamoic Acid SCHEMBL517502 0.95 SLC6A4 (0.51) SLC6A4MAPTHRH1LMNAADORA3
Pamoic Acid SCHEMBL16222836 0.93 SLC6A4 (0.63) SLC6A4MAPTHRH1LMNAADORA3
Pamoic Acid SCHEMBL517584 0.92 SLC6A4 (0.47) SLC6A4MAPTHRH1LMNAADORA3
Imipramine SCHEMBL518586 0.88 KMT2A (0.44) SLC6A4MAPTHRH1LMNAADORA3
Imipramine SCHEMBL2098515 0.84 LMNA (0.62) SLC6A4MAPTHRH1LMNAADORA3
Pamoic Acid SCHEMBL15533092 0.83 SLC6A4 (0.48) SLC6A4MAPTHRH1LMNAADORA3
SCHEMBL5608291 0.82 SLC6A4 (0.47) SLC6A4MAPTHRH1LMNAADORA3
Imipramine SCHEMBL4283852 0.80 SLC6A4 (0.71) SLC6A4MAPTHRH1LMNAADORA3
Imipramine SCHEMBL20644144 0.77 SLC6A4 (0.83) SLC6A4MAPTHRH1LMNAADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1181 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025024501-A1 NEUROMODULATORY PEPTIDES LACTOCORE, INC. (US) 2025-01-30 WO claimed
CN-113573723-B Synthetic neuromodulatory peptides 拉托科公司 2024-12-03 CN claimed
US-20240282425-A1 AUTHENTICATION METHODS AND SYSTEMS FOR DISPENSED PRESCRIPTIONS LOW GORDON KEITH (US) 2024-08-22 US claimed
US-20230248737-A1 COMPOSITIONS AND METHODS FOR TREATING PSYCHIATRIC DISORDERS OR SYMPTOMS THEREOF PSYRX LTD. (IL) 2023-08-10 US claimed
EP-4175643-A1 COMPOSITIONS AND METHODS FOR TREATING PSYCHIATRIC DISORDERS OR SYMPTOMS THEREOF Psyrx Ltd. (IL) 2023-05-10 EP claimed
US-20230140798-A1 SYNTHETIC PEPTIDES DIRECTED AGAINST THE METABOTROPIC GLUTAMATE RECEPTOR 5 LACTOCORE INC (US) 2023-05-04 US claimed
EP-4135741-A1 SYNTHETIC PEPTIDES FOR MODULATING THE METABOTROPIC GLUTAMATE RECEPTOR 5 Lactocore, Inc. (US) 2023-02-22 EP claimed
CN-115379847-A Synthetic peptides for modulating metabotropic glutamate receptor 5 拉托科公司 2022-11-22 CN claimed
US-20220175873-A1 SYNTHETIC NEUROMODULATORY PEPTIDES LACTOCORE, INC. 2022-06-09 US claimed
EP-3938375-A2 SYNTHETIC NEUROMODULATORY PEPTIDES Lactocore, Inc. (US) 2022-01-19 EP claimed
US-20060148785-A1 Medicine for treating gastrointestinal disorder including fecal incontinence LUNDEEN JAMES E 2006-07-06 US claimed
US-20060148781-A1 Method and medicine for treating gastrointestinal disorder in a non-human mammal SIR ISAAC NEWTON ENTERPRISES LLC 2006-07-06 US claimed
US-20050113365-A1 Method and medicine for treating gastrointestinal disorder including irritable bowel syndrome SIR ISAAC NEWTON ENTERPRISES LLC (US) 2005-05-26 US claimed
WO-2004100899-A2 USE OF SECRETIN IN TREATMENTS OF DISORDERS ASSOCIATED WITH THE AMYGDALA THE MCLEAN HOSPITAL CORPORATION (US) 2004-11-25 WO claimed
US-20030139698-A1 Medicated wrap HYSON MORTON I (US) 2003-07-24 US claimed
EP-1309301-A1 MEDICATED WRAP Hyson, Morton I. (US) 2003-05-14 EP claimed
US-20020035105-A1 Composition and method combining an antidepressant with an NMDA receptor antagonist, for treating neuropathic pain ENDO PHARMACEUTICALS INC. 2002-03-21 US claimed
WO-2001080797-A1 MEDICATED WRAP HYSON MORTON I (US) 2001-11-01 WO claimed
EP-0980247-A1 COMPOSITION AND METHOD COMBINING AN ANTIDEPRESSANT WITH AN NMDA RECEPTOR ANTAGONIST, FOR TREATING NEUROPATHIC PAIN Algos Pharmaceutical Corporation (US) 2000-02-23 EP claimed
WO-1998050044-A1 COMPOSITION AND METHOD COMBINING AN ANTIDEPRESSANT WITH AN NMDA RECEPTOR ANTAGONIST, FOR TREATING NEUROPATHIC PAIN ALGOS PHARMACEUTICAL CORPORATION (US) 1998-11-12 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050113365-A1 Method and medicine for treating gastrointestinal disorder including irritable bowel syndrome SI, TPH1, FABP2 SLC6A4 27/4885HRH1 42/4885DRD2 71/4885
US-20230248737-A1 COMPOSITIONS AND METHODS FOR TREATING PSYCHIATRIC DISORDERS OR SYMPTOMS THEREOF GRIN2C, HTR5A, HTR2A SLC6A4 72/4885HRH1 923/4885DRD2 32/4885
US-20060148785-A1 Medicine for treating gastrointestinal disorder including fecal incontinence SI, SLC10A2, HNMT SLC6A4 21/4885HRH1 272/4885DRD2 586/4885
US-20060148781-A1 Method and medicine for treating gastrointestinal disorder in a non-human mammal SI, FABP2, FABP6 SLC6A4 24/4885HRH1 69/4885DRD2 259/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.