SCHEMBL4112185

SCHEMBL4112185

CC(C(O)c1ccccc1)N(C)C(=O)Oc1cnc(NCc2ccccn2)nc1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 6/20 0.44
VNN1 O95497 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
GAA P10253 1/20 0.38
CCNA2 P20248 2/20 0.38
CDK2 P24941 2/20 0.38
CCNA1 P78396 2/20 0.38
AURKA O14965 1/20 0.38
MAOB P27338 1/20 0.37
KCNH2 Q12809 1/20 0.36
NPY2R P49146 1/20 0.36
NAMPT P43490 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
SYK P43405 1/20 0.36
AURKB Q96GD4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3943937 0.89 NPY5R (0.47) NPY5RVNN1GAANPY2R
SCHEMBL3946248 0.84 NPY5R (0.42) NPY5RHDAC3HDAC1HDAC2HDAC6
SCHEMBL3951253 0.77 NPY5R (0.46) NPY5RGAANPY2R
SCHEMBL1383650 0.75 LMNA (0.43) HDAC3HDAC1HDAC2HDAC6CCNA2
SCHEMBL3442663 0.71 HDAC3 (0.52) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL3946609 0.67 NPY5R (0.43) NPY5RGAA
SCHEMBL3948201 0.66 SLC6A2 (0.37) LMNASYKAURKBINCENP
SCHEMBL3942976 0.66 CASR (0.41) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL3390661 0.66 GAA (0.54) NPY5RGAANPY2RKDM4ELMNA
SCHEMBL13819023 0.66 GAA (0.54) NPY5RGAANPY2RKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718632-B1 PYRIMIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS SANOFI AVENTIS (FR) 2009-04-22 EP claimed