SCHEMBL4149156

SCHEMBL4149156

CC(C)(C)OC(=O)n1cc2ccc(CO)cc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 1/20 0.40
NR1H2 P55055 9/20 0.39
NR1H3 Q13133 3/20 0.36
CA12 O43570 3/20 0.36
CA2 P00918 3/20 0.36
CA3 P07451 3/20 0.36
CA6 P23280 3/20 0.36
CA7 P43166 3/20 0.36
CA9 Q16790 3/20 0.36
CA14 Q9ULX7 3/20 0.36
CA5B Q9Y2D0 3/20 0.36
CA5A P35218 2/20 0.36
CA4 P22748 2/20 0.36
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
PTGS1 P23219 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
CYP4F2 P78329 1/20 0.34
CYP4A11 Q02928 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16041668 0.87 NR1H2 (0.48) GPR119NR1H2NR1H3CA12CA2
SCHEMBL17242214 0.87 NR1H2 (0.38) GPR119NR1H2NR1H3PTGS1AKR1C3
SCHEMBL23727382 0.85 NR1H2 (0.36) GPR119NR1H2NR1H3PTGS1AKR1C3
SCHEMBL15878871 0.81 GPR119 (0.37) GPR119NR1H2
SCHEMBL22980683 0.80 HDAC8 (0.36) NR1H2NR1H3PTGS1AKR1C3AKR1C2
SCHEMBL17965623 0.80 ESR2 (0.46) NR1H2MEN1KMT2A
SCHEMBL15878939 0.79 CHKA (0.47) MEN1KMT2AHDAC6KDM4ELMNA
SCHEMBL1394177 0.79 NR1H2 (0.47) NR1H2NR1H3MEN1KMT2AKDM4E
SCHEMBL2144869 0.79 USP30 (0.40) NR1H2HDAC1NPC1LMNAMAPT
SCHEMBL2143961 0.79 GABRG2 (0.41) GPR119NR1H2NR1H3SETD7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12570642-B2 GLP-IR modulating compounds GILEAD SCIENCES, INC. (US) 2026-03-10 US disclosed
EP-4691554-A2 GLP-1R MODULATING COMPOUNDS Gilead Sciences, Inc. (US) 2026-02-11 EP disclosed
US-12517130-B2 Isoindoline derivatives which bind to an ATP binding site Neophore Limited (GB) 2026-01-06 US disclosed
EP-4271672-B1 CARBOXY-BENZIMIDAZOLE GLP-1R MODULATING COMPOUNDS GILEAD SCIENCES INC (US) 2025-12-03 EP disclosed
EP-4506344-A1 1,4-DIHETEROCYCLIC SUBSTITUTED AROMATIC RING OR AROMATIC HETEROCYCLIC COMPOUND AND USE THEREOF Bebetter Med Inc. (CN) 2025-02-12 EP disclosed
US-20240293392-A1 INHIBITOR COMPOUNDS Neophore Limited (GB) 2024-09-05 US disclosed
WO-2024173646-A1 CYCLIN-DEPENDENT KINASE DEGRADING COMPOUNDS INNOVO THERAPEUTICS, INC. (US) 2024-08-22 WO disclosed
US-20240199589-A1 GLP-1R MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2024-06-20 US disclosed
EP-4373819-A1 INHIBITOR COMPOUNDS Neophore Limited (GB) 2024-05-29 EP disclosed
US-11858918-B2 GLP-1R modulating compounds GILEAD SCIENCES, INC. (US) 2024-01-02 US disclosed
US-11267826-B2 Penicillin-binding protein inhibitors VenatoRx Pharmaceuticals, Inc. (US) 2022-03-08 US disclosed
WO-2021229152-A1 CYP11A1 INHIBITORS ORION CORPORATION (FI) 2021-11-18 WO disclosed
WO-2021148786-A1 ISOINDOLINE DERIVATIVES WHICH BIND TO AN ATP BINDING SITE Neophore Limited (GB) 2021-07-29 WO disclosed
EP-3630783-A1 PENICILLIN-BINDING PROTEIN INHIBITORS Venatorx Pharmaceuticals, Inc. (US) 2020-04-08 EP disclosed
US-20200102331-A1 PENICILLIN-BINDING PROTEIN INHIBITORS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2020-04-02 US disclosed
WO-2018218154-A1 PENICILLIN-BINDING PROTEIN INHIBITORS VenatoRx Pharmaceuticals, Inc. (US) 2018-11-29 WO disclosed
US-20160090364-A1 PHTHALAZINONES AND ISOQUINOLINONES AS ROCK INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2016-03-31 US disclosed
US-9221767-B2 Substituted phthalazinones as rock inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2015-12-29 US disclosed
US-20140206686-A1 PHTHALAZINONES AND ISOQUINOLINONES AS ROCK INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2014-07-24 US disclosed
US-20090215742-A1 AMIDE RESORCINOL COMPOUNDS PFIZER, INC. 2009-08-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140206686-A1 PHTHALAZINONES AND ISOQUINOLINONES AS ROCK INHIBITORS MYLK, MYLK2, ROCK1 GPR119 1862/4885NR1H2 1671/4885NR1H3 2014/4885
US-11267826-B2 Penicillin-binding protein inhibitors PEPD, BPGM, EBPL GPR119 3556/4885NR1H2 4732/4885NR1H3 4783/4885
US-20160090364-A1 PHTHALAZINONES AND ISOQUINOLINONES AS ROCK INHIBITORS MYLK, MYLK2, ROCK1 GPR119 1862/4885NR1H2 1671/4885NR1H3 2014/4885
US-20240293392-A1 INHIBITOR COMPOUNDS MSH2, PMS2, MSH6 GPR119 2087/4885NR1H2 2027/4885NR1H3 2514/4885
US-20090215742-A1 AMIDE RESORCINOL COMPOUNDS HSP90AB1, HSP90AA1, HSP90AB2P GPR119 1904/4885NR1H2 90/4885NR1H3 144/4885
US-20200102331-A1 PENICILLIN-BINDING PROTEIN INHIBITORS PEPD, BPGM, EBPL GPR119 3556/4885NR1H2 4732/4885NR1H3 4783/4885
US-11858918-B2 GLP-1R modulating compounds GLP1R, GIPR, GPR119 GPR119 3/4885NR1H2 486/4885NR1H3 812/4885
US-20240199589-A1 GLP-1R MODULATING COMPOUNDS GLP1R, GIPR, GPR119 GPR119 3/4885NR1H2 486/4885NR1H3 812/4885
US-12570642-B2 GLP-IR modulating compounds GLP1R, GIPR, GPR119 GPR119 3/4885NR1H2 188/4885NR1H3 269/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.