Iodide

Iodide

SCHEMBL4155309

C[N+]1(C)CCN(C(=O)Nc2cc(F)cc(F)c2)CC1.[I-]

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 5/20 0.47
ALDH1A1 P00352 4/20 0.47
CYP2D6 P10635 3/20 0.47
KMT2A Q03164 1/20 0.45
CYP2C19 P33261 2/20 0.45
CYP1A2 P05177 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.43
USP2 O75604 2/20 0.43
POLB P06746 1/20 0.43
MAPT P10636 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
S1PR2 O95136 2/20 0.43
CYP2C9 P11712 1/20 0.43
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL4166734 0.86 CYP2D6 (0.65) ALDH1A1CYP2D6CYP2C19CYP1A2SMN1; SMN2
Iodide SCHEMBL4160980 0.84 CACNA1H (0.42) CACNA1HALDH1A1CYP2D6KMT2ACYP2C19
Iodide SCHEMBL4173002 0.83 RAB9A (0.51) ALDH1A1USP2POLBMAPTNPSR1
Iodide SCHEMBL4155962 0.82 NPSR1 (0.67) ALDH1A1KMT2APOLBMAPTNPSR1
Iodide SCHEMBL4154016 0.82 CACNA1H (0.41) CACNA1HALDH1A1CYP2D6KMT2ACYP2C19
SCHEMBL4303277 0.80 KDM4E (0.58) CACNA1HALDH1A1CYP2D6KMT2ASMN1; SMN2
Iodide SCHEMBL4154030 0.77 NPSR1 (0.68) ALDH1A1KMT2ASMN1; SMN2POLBMAPT
Iodide SCHEMBL4159269 0.74 ALDH1A1 (0.70) ALDH1A1KMT2ASMN1; SMN2USP2MAPT
Iodide SCHEMBL4162697 0.74 TRPV1 (0.57) ALDH1A1KMT2APOLBMAPTNPSR1
SCHEMBL4301848 0.74 CACNA1H (0.48) CACNA1HALDH1A1MAPTNPSR1S1PR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090118303-A1 SEROTONIN 5-HT3 RECEPTOR AGONIST RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2009-05-07 US disclosed
US-7485646-B2 Serotonin 5-HT3 receptor agonist RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2009-02-03 US disclosed
US-20070265277-A1 Serotonin 5-Ht3 Receptor Agonist RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2007-11-15 US disclosed
EP-1798227-A1 SEROTONIN 5-HT3 RECEPTOR AGONIST Research Foundation Itsuu Laboratory (JP) 2007-06-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090118303-A1 SEROTONIN 5-HT3 RECEPTOR AGONIST HTR3A, HTR7, HTR1A CACNA1H 794/4885ALDH1A1 2805/4885CYP2D6 1577/4885
US-20070265277-A1 Serotonin 5-Ht3 Receptor Agonist HTR3A, HTR7, HTR1A CACNA1H 794/4885ALDH1A1 2805/4885CYP2D6 1577/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.