SCHEMBL4156587

SCHEMBL4156587

CCc1c(O)cccc1-c1cc[nH]n1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
GFER P55789 1/20 0.33
IDO1 P14902 1/20 0.33
DAO P14920 1/20 0.33
ALOX15 P16050 4/20 0.32
NFKB1 P19838 3/20 0.32
RAB9A P51151 3/20 0.32
NFKB2 Q00653 3/20 0.32
RELA Q04206 3/20 0.32
MAPT P10636 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
TSHR P16473 2/20 0.32
USP2 O75604 1/20 0.32
HPGD P15428 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL206363 0.77 IDO1 (0.53) ALDH1A1IDO1ALOX15NFKB1RAB9A
SCHEMBL16527875 0.76 GABRA1 (0.42) ALDH1A1IDO1ALOX15NFKB1RAB9A
SCHEMBL5527507 0.75 IDO1 (0.34) IDO1ALOX15NFKB1NFKB2RELA
SCHEMBL4156586 0.74 DAO (0.42) DAOCA12CA1CA2CA7
SCHEMBL11620477 0.73 TRPA1 (0.39) IDO1MAPT
SCHEMBL23923799 0.71 APP (0.40) ALDH1A1IDO1DAOALOX15NFKB1
SCHEMBL28059620 0.71 ALDH1A1 (0.43) ALDH1A1GFERIDO1ALOX15NFKB1
SCHEMBL27506231 0.71 TRPA1 (0.47) ALDH1A1IDO1DAOALOX15RAB9A
SCHEMBL21375829 0.70 ADRA2A (0.34) ALDH1A1DAOALOX15RAB9AMAPT
SCHEMBL68691 0.70 GABRA1 (0.48) ALDH1A1ALOX15NFKB1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044063-A1 PYRIMIDINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER Astra Zeneca AB (SE) 2009-04-08 EP disclosed
WO-2008001070-A1 PYRIMIDINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2008-01-03 WO disclosed