Omaciclovir

Omaciclovir

SCHEMBL417577

Nc1nc2c(ncn2CC(CO)CCO)c(=O)[nH]1

nearest known ligand 0.76

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TK1 P04183 2/20 0.62
BLM P54132 2/20 0.62
MEN1 O00255 1/20 0.62
ALDH1A1 P00352 1/20 0.62
LMNA P02545 1/20 0.62
CYP3A4 P08684 1/20 0.62
NFKB1 P19838 1/20 0.62
VCP P55072 1/20 0.62
KMT2A Q03164 1/20 0.62
SMN1; SMN2 Q16637 1/20 0.62
HIF1A Q16665 1/20 0.62
PNP P00491 2/20 0.61
USP2 O75604 1/20 0.61
TSHR P16473 1/20 0.61
EDNRA P25101 1/20 0.61
HTR2A P28223 1/20 0.61
RECQL P46063 1/20 0.61
HBB P68871 1/20 0.61
HSD17B10 Q99714 1/20 0.61
HPRT1 P00492 12/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Omaciclovir SCHEMBL712427 1.00 TK1 (0.62) TK1BLMMEN1ALDH1A1LMNA
Omaciclovir SCHEMBL10507800 0.99 TK1 (0.61) TK1BLMMEN1ALDH1A1LMNA
Omaciclovir SCHEMBL571367 0.95 HPRT1 (0.66) TK1BLMMEN1ALDH1A1LMNA
SCHEMBL10506595 0.95 TK1 (0.65) TK1BLMMEN1ALDH1A1LMNA
Tiviciclovir SCHEMBL6944256 0.92 BLM (0.67) TK1BLMMEN1ALDH1A1LMNA
Omaciclovir SCHEMBL9430446 0.92 TK1 (0.55) TK1BLMMEN1ALDH1A1LMNA
Tiviciclovir SCHEMBL7745021 0.91 BLM (0.66) TK1BLMMEN1ALDH1A1LMNA
SCHEMBL10507335 0.91 TK1 (0.67) TK1BLMMEN1ALDH1A1LMNA
SCHEMBL16488939 0.91 TK1 (0.60) TK1BLMMEN1ALDH1A1LMNA
SCHEMBL10509880 0.90 TK1 (0.69) TK1BLMMEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 391 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160346287-A1 METHOD OF TREATING VIRAL INFECTIONS EPIPHANY BIOSCIENCES, INC. 2016-12-01 US claimed
US-20150050241-A1 METHOD OF TREATING VIRAL INFECTIONS EPIPHANY BIOSCIENCES, INC. 2015-02-19 US claimed
WO-2014047562-A2 METHOD OF TREATING AND/OR PREVENTING SHINGLES AND METHOD OF TREATING AND/OR PREVENTING ZOSTER ASSOCIATED PAIN EPIPHANY BIOSCIENCES (US) 2014-03-27 WO claimed
EP-1720856-B1 HIV INTEGRASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2013-08-14 EP claimed
US-8455497-B2 Inhibitors of aspartyl protease VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-06-04 US claimed
EP-1686113-B1 Inhibitors of aspartyl protease VERTEX PHARMA (US) 2011-11-23 EP claimed
JP-4503896-B2 2010-07-14 JP claimed
US-20090274650-A1 INHIBITORS OF ASPARTYL PROTEASE VERTEX PHARMACEUTICALS INCORPORATED 2009-11-05 US claimed
WO-2009120358-A1 OLIGOMER-NITROGENOUS BASE CONJUGATES NEKTAR THERAPEUTICS (US) 2009-10-01 WO claimed
US-20090053172-A1 HETEROCYCLIC COMPOUNDS AS CCR5 ANTAGONISTS AQUINO CHRISTOPHER JOSEPH 2009-02-26 US claimed
WO-2000076961-A1 INHIBITORS OF ASPARTYL PROTEASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2000-12-21 WO claimed
WO-2000029027-A1 ANTIVIRAL FORMULATIONS COMPRISING PROPYLENE GLYCOL AND AN ISOPROPYL ALKANOIC ACID ESTER MEDIVIR AB (SE) 2000-05-25 WO claimed
EP-0942916-A2 NUCLEOSIDES Medivir Aktiebolag (SE) 1999-09-22 EP claimed
WO-1998021223-A1 NUCLEOSIDES MEDIVIR AB (SE) 1998-05-22 WO claimed
WO-1996022098-A1 USE OF ACYCLIC PURINE DERIVATIVES FOR TREATING RESTENOSIS THE WELLCOME FOUNDATION LIMITED (GB) 1996-07-25 WO claimed
EP-0165289-B1 NOVEL DERIVATIVES OF GUANINE Medivir Aktiebolag (SE) 1989-04-05 EP claimed
US-4798833-A VIRICIDES ASTRA LAKEMEDEL AKTIEBOLAG (SE) 1989-01-17 US claimed
EP-0165289-A1 NOVEL DERIVATIVES OF GUANINE. ASTRA LAEKEMEDEL AB (SE) 1985-12-27 EP claimed
WO-1985002845-A1 NOVEL DERIVATIVES OF GUANINE Astra Läkemedel Aktiebolag (SE) 1985-07-04 WO claimed
EP-0146516-A2 Derivatives of Guanine, process for their preparation and a pharmaceutical preparation Astra Läkemedel Aktiebolag (SE) 1985-06-26 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160346287-A1 METHOD OF TREATING VIRAL INFECTIONS IFNG, BCL9, GDA TK1 337/4885BLM 37/4885MEN1 74/4885
US-20090053172-A1 HETEROCYCLIC COMPOUNDS AS CCR5 ANTAGONISTS CCR5, CXCR3, CCR1 TK1 297/4885BLM 3729/4885MEN1 4508/4885
US-20150050241-A1 METHOD OF TREATING VIRAL INFECTIONS IFNG, BCL9, GDA TK1 337/4885BLM 37/4885MEN1 74/4885
US-20090274650-A1 INHIBITORS OF ASPARTYL PROTEASE SPINT2, DNPEP, PRSS1 TK1 2033/4885BLM 4822/4885MEN1 4418/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.