Omaciclovir

Omaciclovir

SCHEMBL712427

Nc1nc2c(ncn2C[C@H](CO)CCO)c(=O)[nH]1

nearest known ligand 0.76

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TK1 P04183 2/20 0.62
BLM P54132 2/20 0.62
MEN1 O00255 1/20 0.62
ALDH1A1 P00352 1/20 0.62
LMNA P02545 1/20 0.62
CYP3A4 P08684 1/20 0.62
NFKB1 P19838 1/20 0.62
VCP P55072 1/20 0.62
KMT2A Q03164 1/20 0.62
SMN1; SMN2 Q16637 1/20 0.62
HIF1A Q16665 1/20 0.62
PNP P00491 2/20 0.61
USP2 O75604 1/20 0.61
TSHR P16473 1/20 0.61
EDNRA P25101 1/20 0.61
HTR2A P28223 1/20 0.61
RECQL P46063 1/20 0.61
HBB P68871 1/20 0.61
HSD17B10 Q99714 1/20 0.61
HPRT1 P00492 12/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Omaciclovir SCHEMBL417577 1.00 TK1 (0.62) TK1BLMMEN1ALDH1A1LMNA
Omaciclovir SCHEMBL10507800 0.99 TK1 (0.61) TK1BLMMEN1ALDH1A1LMNA
Omaciclovir SCHEMBL571367 0.95 HPRT1 (0.66) TK1BLMMEN1ALDH1A1LMNA
SCHEMBL10506595 0.95 TK1 (0.65) TK1BLMMEN1ALDH1A1LMNA
Tiviciclovir SCHEMBL6944256 0.92 BLM (0.67) TK1BLMMEN1ALDH1A1LMNA
Omaciclovir SCHEMBL9430446 0.92 TK1 (0.55) TK1BLMMEN1ALDH1A1LMNA
Tiviciclovir SCHEMBL7745021 0.91 BLM (0.66) TK1BLMMEN1ALDH1A1LMNA
SCHEMBL10507335 0.91 TK1 (0.67) TK1BLMMEN1ALDH1A1LMNA
SCHEMBL16488939 0.91 TK1 (0.60) TK1BLMMEN1ALDH1A1LMNA
SCHEMBL10509880 0.90 TK1 (0.69) TK1BLMMEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 88 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024167952-A1 OXIDATIVELY CLEAVABLE ORGANOPHOSPHATE DRUGS UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2024-08-15 WO claimed
WO-2024118480-A1 USE OF ANTIVIRAL AGENTS, COMPOSITION OF MATTER, COMBINATION PREPARATIONS/AGENTS TO TREAT CHRONIC DISEASES ASSOCIATED WITH EPSTEIN-BARR VIRUS AND OTHER HUMAN HERPES VIRUSES EPIPHANY BIOSCIENCES (US) 2024-06-06 WO claimed
US-20230158000-A1 PHARMACEUTICAL COMPOSITION FOR TREATING OR PREVENTING VIRAL HEPATITIS AND THE USE THEREOF HOLY HAID LAB CORP (CN) 2023-05-25 US claimed
WO-2014047562-A2 METHOD OF TREATING AND/OR PREVENTING SHINGLES AND METHOD OF TREATING AND/OR PREVENTING ZOSTER ASSOCIATED PAIN EPIPHANY BIOSCIENCES (US) 2014-03-27 WO claimed
EP-2841109-B1 PRODRUGS OF HYDROXYL-COMPRISING DRUGS ASCENDIS PHARMA AS (DK) 2026-04-15 EP disclosed
CN-121401266-A Application of omalovir in inhibiting influenza A virus 福建农林大学 2026-01-27 CN disclosed
US-20250387363-A1 LIQUID EPINEPHRINE PRODRUG FORMULATIONS AND LIQUID EPINEPHRINE FORMULATIONS INSIGNIS THERAPEUTICS INC (US) 2025-12-25 US disclosed
EP-3782649-B1 BIODEGRADABLE POLYETHYLENE GLYCOL BASED WATER-INSOLUBLE HYDROGELS ASCENDIS PHARMA AS (DK) 2025-05-14 EP disclosed
US-20250000821-A1 METHODS OF USING DIPIVEFRIN Insignis Therapeutics, Inc. 2025-01-02 US disclosed
WO-2024174020-A1 HERPES ZOSTER TREATMENT XBIOTECH INC. (CA) 2024-08-29 WO disclosed
WO-2024163327-A1 EPSTEIN-BARR VIRUS GLYCOPROTEIN 42 IMMUNOGENS FOR VACCINATION AND ANTIBODY DISCOVERY THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2024-08-08 WO disclosed
WO-2024118480-A1 USE OF ANTIVIRAL AGENTS, COMPOSITION OF MATTER, COMBINATION PREPARATIONS/AGENTS TO TREAT CHRONIC DISEASES ASSOCIATED WITH EPSTEIN-BARR VIRUS AND OTHER HUMAN HERPES VIRUSES EPIPHANY BIOSCIENCES (US) 2024-06-06 WO disclosed
US-5869493-A ANTIVIRALS AGAINST HERPES AND RETROVIRUSES MEDIVIR AB (SE) 1999-02-09 US disclosed
EP-0888348-A1 ACYCLIC NUCLEOSIDE DERIVATIVES Medivir Aktiebolag (SE) 1999-01-07 EP disclosed
EP-0880521-A1 SYNTHESIS OF ACYCLIC NUCLEOSIDES Medivir Aktiebolag (SE) 1998-12-02 EP disclosed
WO-1998034917-A2 SYNTHESIS OF ACYCLIC NUCLEOSIDE DERIVATIVES MEDIVIR AB (SE) 1998-08-13 WO disclosed
WO-1997030052-A1 SYNTHESIS OF ACYCLIC NUCLEOSIDES MEDIVIR AB (SE) 1997-08-21 WO disclosed
WO-1997030051-A1 ACYCLIC NUCLEOSIDE DERIVATIVES MEDIVIR AB (SE) 1997-08-21 WO disclosed
WO-1995007910-A1 ANTIVIRAL INDOLE DERIVATIVES THE WELLCOME FOUNDATION LIMITED (GB) 1995-03-23 WO disclosed
WO-1995005179-A1 THERAPEUTIC COMBINATION CONTAINING AN ANTI-VARICELLA ZOSTER VIRUS COMPOUND AND LAMOTRIGINE THE WELLCOME FOUNDATION LIMITED (GB) 1995-02-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230158000-A1 PHARMACEUTICAL COMPOSITION FOR TREATING OR PREVENTING VIRAL HEPATITIS AND THE USE THEREOF SLC10A1, HAVCR2, SLC10A2 TK1 2014/4885BLM 780/4885MEN1 1304/4885
US-20250000821-A1 METHODS OF USING DIPIVEFRIN QDPR, DNPEP, DPEP1 TK1 2109/4885BLM 1124/4885MEN1 419/4885
US-20250387363-A1 LIQUID EPINEPHRINE PRODRUG FORMULATIONS AND LIQUID EPINEPHRINE FORMULATIONS ADRB3, ADRB2, ADRB1 TK1 3492/4885BLM 1987/4885MEN1 1013/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.