SCHEMBL419198

SCHEMBL419198

CSc1c(C(F)(F)C(F)(F)F)ccc(C(=O)O)c1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 1/20 0.35
PKM P14618 1/20 0.35
LIG1 P18858 1/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
HAAO P46952 1/20 0.34
MCL1 Q07820 1/20 0.33
NOTUM Q6P988 3/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
CYP1A2 P05177 1/20 0.32
SORT1 Q99523 2/20 0.32
USP2 O75604 1/20 0.32
CYP2C19 P33261 1/20 0.32
ASPH Q12797 1/20 0.32
TSHR P16473 1/20 0.32
DAO P14920 1/20 0.32
DHODH Q02127 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL412257 0.89 TAS2R14 (0.42) TAS2R14PKMLIG1RXRARXRB
SCHEMBL416274 0.85 CFTR (0.38) PKMLIG1NOTUMALDH1A1KDM4E
SCHEMBL417766 0.78 TAS2R14 (0.38) TAS2R14RXRARXRBHAAONOTUM
SCHEMBL17396421 0.75 HAAO (0.40) RXRBHAAOMCL1NOTUMALDH1A1
SCHEMBL17593679 0.73 KDM4E (0.43) PKMMCL1ALDH1A1KDM4EHPGD
SCHEMBL17395308 0.73 GPR35 (0.40) HAAOMCL1ALDH1A1HPGDHSD17B10
SCHEMBL8726320 0.73 ALDH1A1 (0.41) MCL1NOTUMALDH1A1KDM4EHPGD
SCHEMBL976616 0.72 NOTUM (0.39) TAS2R14PKMLIG1RXRARXRB
SCHEMBL1230305 0.72 NOTUM (0.39) TAS2R14PKMLIG1RXRARXRB
SCHEMBL31440663 0.72 NOTUM (0.39) TAS2R14PKMLIG1RXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595955-B1 (4-HALOGENALKYL-3-THIOBENZOYL)CYCLOHEXANEDIONES AND USE THEREOF AS HERBICIDES BAYER IP GMBH (DE) 2016-11-30 EP disclosed
EP-2595963-B1 4-(4-HALOGENALKYL-3-THIOBENZOYL)PYRAZOLES AND USE THEREOF AS HERBICIDES BAYER IP GMBH (DE) 2014-11-12 EP disclosed
US-8603947-B2 (4-haloalkyl-3-thiobenzoyl)cyclohexanediones and use thereof as herbicides BAYER CROPSCIENCE AG (DE) 2013-12-10 US disclosed
US-8536097-B2 4-(4-haloalkyl-3-thiobenzoyl)pyrazoles and use thereof as herbicides BAYER CROPSCIENCE AG (DE) 2013-09-17 US disclosed
EP-2595963-A1 4-(4-HALOGENALKYL-3-THIOBENZOYL)PYRAZOLES AND USE THEREOF AS HERBICIDES Bayer Intellectual Property GmbH (DE) 2013-05-29 EP disclosed
EP-2595955-A1 (4-HALOGENALKYL-3-THIOBENZOYL)CYCLOHEXANEDIONES AND USE THEREOF AS HERBICIDES Bayer Intellectual Property GmbH (DE) 2013-05-29 EP disclosed
US-20120021904-A1 (4-HALOALKYL-3-THIOBENZOYL)CYCLOHEXANEDIONES AND USE THEREOF AS HERBICIDES BAYER CROPSCIENCE AG (DE) 2012-01-26 US disclosed
US-20120021903-A1 4-(4-HALOALKYL-3-THIOBENZOYL)PYRAZOLES AND USE THEREOF AS HERBICIDES BAYER CROPSCIENCE AG (DE) 2012-01-26 US disclosed
WO-2012010575-A1 (4-HALOGENALKYL-3-THIOBENZOYL)CYCLOHEXANEDIONES AND USE THEREOF AS HERBICIDES BAYER CROPSCIENCE AG (DE) 2012-01-26 WO disclosed
WO-2012010573-A1 4-(4-HALOGENALKYL-3-THIOBENZOYL)PYRAZOLES AND USE THEREOF AS HERBICIDES BAYER CROPSCIENCE AG (DE) 2012-01-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120021904-A1 (4-HALOALKYL-3-THIOBENZOYL)CYCLOHEXANEDIONES AND USE THEREOF AS HERBICIDES CBR3, CBR1, CYP8B1 TAS2R14 1504/4885PKM 2791/4885LIG1 2247/4885
US-20120021903-A1 4-(4-HALOALKYL-3-THIOBENZOYL)PYRAZOLES AND USE THEREOF AS HERBICIDES CBR3, CYP4X1, PRDX4 TAS2R14 954/4885PKM 1345/4885LIG1 1657/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.