SCHEMBL4197282

SCHEMBL4197282

N#CCC1C=CN=C(NCC(O)c2ccccc2)N1c1nc2ccccc2s1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.48
MAPK1 P28482 1/20 0.48
CTSS P25774 4/20 0.34
CTSK P43235 4/20 0.34
CTSL P07711 3/20 0.34
CTSB P07858 3/20 0.34
FAAH O00519 1/20 0.32
GAA P10253 1/20 0.32
CSNK1D P48730 2/20 0.32
NCS1 P62166 1/20 0.32
ALDH1A1 P00352 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GSK3B P49841 1/20 0.32
DPP4 P27487 1/20 0.31
CYP2D6 P10635 1/20 0.31
GPBAR1 Q8TDU6 1/20 0.31
CYP26A1 O43174 1/20 0.31
ACACB O00763 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4192273 0.84 MAPK9 (0.39) MAPK1CTSKALDH1A1NPSR1DPP4
SCHEMBL7706938 0.84 KMT2A (0.37) HPGDALDH1A1NPSR1DPP4CYP2D6
SCHEMBL4186367 0.82 ILK (0.37) HPGDGAAALDH1A1NPSR1DPP4
SCHEMBL4192472 0.82 NPC1 (0.46) ALDH1A1CYP2D6
SCHEMBL4187924 0.82 RAB9A (0.36) HPGDMAPK1GAAALDH1A1NPSR1
SCHEMBL6828604 0.81 IDO1 (0.37) MAPK1ALDH1A1NPSR1DPP4CYP2D6
SCHEMBL4199489 0.81 KMT2A (0.37) MAPK1GAAALDH1A1NPSR1DPP4
Acetonitrile SCHEMBL7707679 0.80 RAB9A (0.35) HPGDMAPK1GAAALDH1A1NPSR1
SCHEMBL4197422 0.80 SMN1; SMN2 (0.41) HPGDGAAALDH1A1CYP2D6
SCHEMBL4187935 0.80 ILK (0.38) MAPK1ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2026802-A2 JNK INHIBITORS FOR TREATMENT OF SKIN DISEASES Laboratoires Serono SA (CH) 2009-02-25 EP disclosed
EP-1904181-A2 JNK INHIBITORS FOR THE TREATMENT OF ENDOMETREOSIS LABORATOIRES SERONO S.A. (CH) 2008-04-02 EP disclosed
WO-2007141224-A2 JNK INHIBITORS FOR TREATMENT OF SKIN DISEASES LABORATOIRES SERONO SA (CH) 2007-12-13 WO disclosed
WO-2007011762-A2 JNK INHIBITORS FOR THE TREATMENT OF ENDOMETREOSIS LABORATOIRES SERONO S.A. (CH) 2007-01-25 WO disclosed