SCHEMBL420878

SCHEMBL420878

CCOC(=O)C=CC1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.45
RECQL P46063 1/20 0.43
EPHX1 P07099 1/20 0.43
GPR119 Q8TDV5 6/20 0.42
GAA P10253 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
USP2 O75604 1/20 0.41
MEN1 O00255 2/20 0.41
ALDH1A1 P00352 2/20 0.41
KMT2A Q03164 2/20 0.41
TSHR P16473 1/20 0.41
LMNA P02545 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
DPP4 P27487 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
THRB P10828 1/20 0.40
PTPN2 P17706 1/20 0.40
PTPN1 P18031 1/20 0.40
PTPN6 P29350 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10154186 1.00 HPGD (0.45) HPGDRECQLEPHX1GPR119GAA
SCHEMBL420877 1.00 HPGD (0.45) HPGDRECQLEPHX1GPR119GAA
SCHEMBL23007135 0.92 GPR119 (0.40) HPGDRECQLEPHX1GPR119GAA
SCHEMBL30663169 0.92 GPR119 (0.40) HPGDRECQLEPHX1GPR119GAA
SCHEMBL26619671 0.92 GPR119 (0.40) HPGDRECQLEPHX1GPR119GAA
SCHEMBL23006816 0.92 GPR119 (0.40) HPGDRECQLEPHX1GPR119GAA
SCHEMBL32687569 0.92 GPR119 (0.40) HPGDRECQLEPHX1GPR119GAA
SCHEMBL20128945 0.91 HPGD (0.45) HPGDRECQLEPHX1GPR119GAA
SCHEMBL16482944 0.88 GPR119 (0.45) HPGDRECQLEPHX1GPR119GAA
SCHEMBL16465716 0.88 GPR119 (0.45) HPGDRECQLEPHX1GPR119GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12569564-B2 Spirocyclic MDM2 modulator and uses thereof NEWAVE PHARMACEUTICAL INC. (US) 2026-03-10 US disclosed
US-12503452-B2 Antimicrobial compounds and methods CURZA GLOBAL, LLC (US) 2025-12-23 US disclosed
US-20250073340-A1 SPIROCYCLIC MDM2 MODULATOR AND USES THEREOF NEWAVE PHARMACEUTICAL INC. 2025-03-06 US disclosed
CN-112384509-B Furin inhibitors 葛兰素史密斯克莱知识产权发展有限公司 2024-04-30 CN disclosed
EP-3790871-B1 FURIN INHIBITORS GLAXOSMITHKLINE IP DEV LTD (GB) 2024-01-24 EP disclosed
US-11773078-B2 Furin inhibitors GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2023-10-03 US disclosed
US-20230159491-A1 Antimicrobial Compounds and Methods NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-05-25 US disclosed
US-20220315556-A1 FURIN INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2022-10-06 US disclosed
WO-2022159644-A1 SPIROCYCLIC MDM2 MODULATOR AND USES THEREOF NEWAVE PHARMACEUTICAL INC. (US) 2022-07-28 WO disclosed
EP-3911644-A1 ANTIMICROBIAL COMPOUNDS AND METHODS Curza Global LLC (US) 2021-11-24 EP disclosed
US-20050075499-A1 Tricyclic compounds protein kinase inhibitors for enhancing the efficacy of anti-neoplastic agents and radiation therapy AGOURON PHARMACEUTICALS, INC. 2005-04-07 US disclosed
US-20050065211-A1 Ester derivatives MSD K.K. (JP) 2005-03-24 US disclosed
US-6846835-B2 Treating chronic obstructive pulmonary disease, chronic bronchitis, asthma, chronic respiratory tract obstruction, fibroid lung, pulmonary emphysema or rhinitis BANYU PHARMACEUTICAL CO., LTD. (JP) 2005-01-25 US disclosed
WO-2004063198-A1 DIAZEPINOINDOLE DERIVATIVES AS KINASE INHIBITORS PFIZER INC. (US) 2004-07-29 WO disclosed
US-20040002504-A1 N-(3-(4-substituted-1-piperidinyl)-1-phenylpropyl) substituted sulfonamides as NK-3 receptor antagonists MERCK SHARP & DOHME LTD. (GB) 2004-01-01 US disclosed
US-20030191316-A1 Ester derivatives MSD K.K. (JP) 2003-10-09 US disclosed
EP-1302458-A1 ESTER DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 2003-04-16 EP disclosed
US-6399619-B1 PREVENTION AND TREATMENT OF AIDS AND VIRAL INFECTION BY HIV MERCK & CO., INC. 2002-06-04 US disclosed
US-5607948-A PLATELET AGGREGATION INHIBITORS, BONE RESORPTION INHIBITORS SUMITOMO PHARMACEUTICALS CO., LTD. (JP) 1997-03-04 US disclosed
EP-0706999-A1 NOVEL DIPIPERIDINE DERIVATIVE SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1996-04-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230159491-A1 Antimicrobial Compounds and Methods MPO, NISCH, RPN2 HPGD 1474/4885RECQL 3644/4885EPHX1 4311/4885
US-20040002504-A1 N-(3-(4-substituted-1-piperidinyl)-1-phenylpropyl) substituted sulfonamides as NK-3 receptor antagonists KCNH3, KCNH2, KCNK3 HPGD 4067/4885RECQL 4217/4885EPHX1 3209/4885
US-20220315556-A1 FURIN INHIBITORS FURIN, TGFB1, PCSK7 HPGD 779/4885RECQL 1664/4885EPHX1 424/4885
US-20030191316-A1 Ester derivatives CHRM3, CHRM2, CHRM1 HPGD 3412/4885RECQL 2111/4885EPHX1 1517/4885
US-20050075499-A1 Tricyclic compounds protein kinase inhibitors for enhancing the efficacy of anti-neoplastic agents and radiation therapy CHEK2, CHEK1, CHKA HPGD 2297/4885RECQL 566/4885EPHX1 3527/4885
US-20250073340-A1 SPIROCYCLIC MDM2 MODULATOR AND USES THEREOF FOXM1, MDM2, FOXO1 HPGD 1572/4885RECQL 35/4885EPHX1 3196/4885
US-12569564-B2 Spirocyclic MDM2 modulator and uses thereof MDM2, TP53, XIAP HPGD 2935/4885RECQL 446/4885EPHX1 2954/4885
US-20050065211-A1 Ester derivatives CHRM3, CHRM2, CHRM1 HPGD 2601/4885RECQL 1760/4885EPHX1 1253/4885
US-11773078-B2 Furin inhibitors FURIN, TGFB1, PCSK7 HPGD 779/4885RECQL 1664/4885EPHX1 424/4885
US-12503452-B2 Antimicrobial compounds and methods MPO, NISCH, RPN2 HPGD 1474/4885RECQL 3644/4885EPHX1 4311/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.