SCHEMBL422756

SCHEMBL422756

O=[N+]([O-])c1cc(Br)cnc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.39
MAPK1 P28482 2/20 0.37
TSHR P16473 2/20 0.37
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
PKM P14618 1/20 0.37
KMT2A Q03164 1/20 0.37
EGFR P00533 1/20 0.36
AKR1B1 P15121 1/20 0.36
GPR35 Q9HC97 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
S100A4 P26447 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
PIN1 Q13526 2/20 0.36
ALDH1A1 P00352 2/20 0.35
CYP3A4 P08684 2/20 0.35
TDP1 Q9NUW8 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29445407 0.80 MAPK1 (0.44) MAPK1TSHRPOLBGPR35PIN1
SCHEMBL113455 0.80 MAPK1 (0.44) MAPK1TSHRPOLBGPR35PIN1
SCHEMBL202290 0.80 ERN1 (0.41) ERN1MEN1POLBPKMKMT2A
SCHEMBL29600703 0.80 ERN1 (0.41) ERN1MEN1POLBPKMKMT2A
SCHEMBL6512051 0.80 ERN1 (0.41) ERN1MEN1POLBPKMKMT2A
SCHEMBL5033872 0.80 MAPT (0.42) MAPK1MEN1POLBKMT2AEGFR
SCHEMBL29780392 0.78 AHR (0.51) MAPK1TSHRMEN1PKMKMT2A
SCHEMBL985995 0.78 AHR (0.51) MAPK1TSHRMEN1PKMKMT2A
SCHEMBL27732124 0.78 KMT2A (0.41) ERN1MEN1POLBPKMKMT2A
SCHEMBL18224443 0.77 ATM (0.31) ERN1EGFRS100A4TRPV1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1399 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120887867-B Quinoline biaryl heterocycle PI3K/HDAC double-target small molecule inhibitor and application thereof 浙江中医药大学 2026-05-15 CN claimed
CN-112441970-A 2, 5-disubstituted-3-aminopyridine compound and preparation method and application thereof 天津医科大学 2021-03-05 CN claimed
CN-102372707-A Synthetic method of 6-methyl-4-bromine-1,6-dihydropyrrole[2,3-c]pyridine-7-one WUXI APPTEC CO LTD 2012-03-14 CN claimed
EP-4747248-A1 COMPOUNDS FOR USE IN A METHOD OF TARGETED PROTEIN DEGRADATION Institute of Cancer Research: Royal Cancer Hospital (The) (GB) 2026-05-27 EP disclosed
US-12637467-B2 Inhibitor of BTK and mutants thereof NEWAVE PHARMACEUTICAL INC. (US) 2026-05-26 US disclosed
CN-120887867-B Quinoline biaryl heterocycle PI3K/HDAC double-target small molecule inhibitor and application thereof 浙江中医药大学 2026-05-15 CN disclosed
US-20260103464-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYL-PYRIDINE DERIVATIVES BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 2026-04-16 US disclosed
US-12583866-B2 Pyrido[2,3-b][1,4]oxazines or tetrahydropyrido[2,3-b][1,4]oxazepines as IAP antagonists BEONE MEDICINES I GMBH (CH) 2026-03-24 US disclosed
US-20260070880-A1 DYNAMIN ACTIVATORS WALDEN BIOSCIENCES, INC. (US) 2026-03-12 US disclosed
US-12527737-B2 Pharmaceutical formulations of tropomyosin related kinase (TRK) inhibitors GENZYME CORPORATION (US) 2026-01-20 US disclosed
US-20250388583-A1 COMPOUNDS AND METHOD FOR PKMYT1 INHIBITION ENGINE BIOSCIENCES PTE LTD (SG) 2025-12-25 US disclosed
EP-0107914-B1 AMINOPYRIMIDINONE DERIVATIVES USEFUL AS HISTAMINE H1-ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1986-05-14 EP disclosed
US-4537891-A 2-(3,5-Substituted-2-pyridylalkylamino)-5-benzyl-4-pyrimidones SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1985-08-27 US disclosed
US-4537890-A 2-(3,5-Substituted-2-pyridylalkylamino)-5-oxopyridylmethyl-4-pyrimidones useful as histamine H1 -antagonists SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1985-08-27 US disclosed
US-4532252-A 3,5-Substituted-2-pyridylalkylamino compounds having histamine H1 -antagonist activity SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1985-07-30 US disclosed
EP-0134091-A1 Pyrimidone derivatives SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1985-03-13 EP disclosed
EP-0122109-A2 Preparation of cyano- or aminoalkyl substituted aromatic amines SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1984-10-17 EP disclosed
EP-0115132-A1 Pyrimidone derivatives SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1984-08-08 EP disclosed
EP-0112142-A2 Pyridine derivatives SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1984-06-27 EP disclosed
EP-0107914-A1 Aminopyrimidinone derivatives useful as histamine H1-antagonists SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1984-05-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12583866-B2 Pyrido[2,3-b][1,4]oxazines or tetrahydropyrido[2,3-b][1,4]oxazepines as IAP antagonists BIRC2, BIRC3, BIRC5 ERN1 4118/4885MAPK1 2218/4885TSHR 3597/4885
US-20260070880-A1 DYNAMIN ACTIVATORS DNM1, DNM1L, DNM2 ERN1 2320/4885MAPK1 715/4885TSHR 2846/4885
US-12527737-B2 Pharmaceutical formulations of tropomyosin related kinase (TRK) inhibitors TPM3, TPM4, MATK ERN1 2625/4885MAPK1 526/4885TSHR 570/4885
US-20250388583-A1 COMPOUNDS AND METHOD FOR PKMYT1 INHIBITION PKMYT1, PKN1, PRKCB ERN1 417/4885MAPK1 267/4885TSHR 548/4885
US-12637467-B2 Inhibitor of BTK and mutants thereof BTK, CNKSR1, SYK ERN1 757/4885MAPK1 614/4885TSHR 328/4885
US-20260103464-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYL-PYRIDINE DERIVATIVES CBR3, CYCS, CBR1 ERN1 2053/4885MAPK1 3819/4885TSHR 197/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.