Cyclo(Prolylglycyl)

Cyclo(Prolylglycyl)

SCHEMBL4243772

O=C1NCC(=O)N2CCC[C@H]12

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
KDM4E B2RXH2 4/20 0.48
MAPT P10636 3/20 0.44
GAA P10253 1/20 0.44
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
HPGD P15428 2/20 0.38
ALOX15 P16050 1/20 0.38
HSD17B10 Q99714 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
PARP1 P09874 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
PPIA P62937 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cyclo(Prolylglycyl) SCHEMBL4247464 1.00 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL30768150 1.00 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL21736594 1.00 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTGAAKMT2A
Cyclo(Prolylglycyl) SCHEMBL3016264 1.00 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL21736595 1.00 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL1189351 0.94 ALDH1A1 (0.43) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL3519704 0.94 ALDH1A1 (0.43) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL3519708 0.94 ALDH1A1 (0.43) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL17516644 0.93 KDM4E (0.43) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL464685 0.93 KDM4E (0.43) ALDH1A1KDM4EMAPTGAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3681504-B1 METHODS OF DETECTION USING X-RAY FLUORESCENCE ICAGEN INC (US) 2023-08-23 EP disclosed
US-11573224-B2 Methods of detection using X-ray fluorescence ICAGEN, LLC (US) 2023-02-07 US disclosed
US-11446398-B2 Regulated biocircuit systems OBSIDIAN THERAPEUTICS, INC. (US) 2022-09-20 US disclosed
US-20210254056-A1 IDENTIFICATION AND TARGETED MODULATION OF GENE SIGNALING NETWORKS CAMP4 THERAPEUTICS CORPORATION 2021-08-19 US disclosed
US-10877035-B2 Advanced drug development and manufacturing ICAGEN, LLC (US) 2020-12-29 US disclosed
US-20200278346-A1 METHODS OF DETECTION USING X-RAY FLUORESCENCE ADJACENT ACQUISITION CO., LLC 2020-09-03 US disclosed
EP-3681504-A1 METHODS OF DETECTION USING X-RAY FLUORESCENCE Icagen, Inc. (US) 2020-07-22 EP disclosed
US-20190192691-A1 REGULATED BIOCIRCUIT SYSTEMS OBSIDIAN THERAPEUTICS, INC. 2019-06-27 US disclosed
WO-2019055754-A1 METHODS OF DETECTION USING X-RAY FLUORESCENCE ICAGEN, INC. (US) 2019-03-21 WO disclosed
WO-2018204764-A1 IDENTIFICATION AND TARGETED MODULATION OF GENE SIGNALING NETWORKS CAMP4 THERAPEUTICS CORPORATION (US) 2018-11-08 WO disclosed
US-20090036455-A1 ARYLPIPERAZINE DERIVATIVE AND USE THEREOF AS 5-HT1A RECEPTOR LIGANDS CEPA SCHWARZ PHARMA, S.L. (ES) 2009-02-05 US disclosed
WO-2008127291-A2 ADVANCED DRUG DEVELOPMENT AND MANUFACTURING LOS ALAMOS NATIONAL SECURITY, LLC (US) 2008-10-23 WO disclosed
US-20080220441-A1 Advanced drug development and manufacturing THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2008-09-11 US disclosed
CN-101087610-A Arylpiperazine derivatives and their use as 5-HT1AUse of receptor ligands SCHWARZ PHARMA S L (ES) 2007-12-12 CN disclosed
US-7304064-B2 1-[(indol-3-yl)carbonyl]piperazine derivatives N.V. ORGANON (NL) 2007-12-04 US disclosed
EP-1549637-B1 1- (INDOL-3-YL)CARBONYL PIPERAZINE DERIVATIVES ORGANON NV (NL) 2007-05-02 EP disclosed
EP-1674103-A1 Arylpiperazine derivatives and use thereof as 5-HT1A receptor ligands Cepa Schwarz Pharma s.l. (ES) 2006-06-28 EP disclosed
US-20050250760-A1 1-[(Indol-3-yl)carbonyl]piperazine derivatives MERCK SHARP & DOHME B.V. (NL) 2005-11-10 US disclosed
EP-1549637-A1 1- (INDOL-3-YL)CARBONYL PIPERAZINE DERIVATIVES Akzo Nobel N.V. (NL) 2005-07-06 EP disclosed
WO-2004000832-A1 1-[(INDOL-3-YL)CARBONYL] PIPERAZINE DERIVATIVES AKZO NOBEL N.V. (NL) 2003-12-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050250760-A1 1-[(Indol-3-yl)carbonyl]piperazine derivatives IDO1, OPRL1, OPRK1 ALDH1A1 689/4885KDM4E 1502/4885MAPT 2304/4885
US-20090036455-A1 ARYLPIPERAZINE DERIVATIVE AND USE THEREOF AS 5-HT1A RECEPTOR LIGANDS HTR1A, HTR5A, HTR2C ALDH1A1 671/4885KDM4E 3602/4885MAPT 486/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.