Cyclo(Prolylglycyl)

Cyclo(Prolylglycyl)

SCHEMBL4247464

O=C1NCC(=O)N2CCC[C@@H]12

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
KDM4E B2RXH2 4/20 0.48
MAPT P10636 3/20 0.44
GAA P10253 1/20 0.44
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
HPGD P15428 2/20 0.38
ALOX15 P16050 1/20 0.38
HSD17B10 Q99714 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
PARP1 P09874 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
PPIA P62937 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30768150 1.00 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL21736594 1.00 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTGAAKMT2A
Cyclo(Prolylglycyl) SCHEMBL3016264 1.00 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL21736595 1.00 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTGAAKMT2A
Cyclo(Prolylglycyl) SCHEMBL4243772 1.00 ALDH1A1 (0.48) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL1189351 0.94 ALDH1A1 (0.43) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL3519704 0.94 ALDH1A1 (0.43) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL3519708 0.94 ALDH1A1 (0.43) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL17516644 0.93 KDM4E (0.43) ALDH1A1KDM4EMAPTGAAKMT2A
SCHEMBL464685 0.93 KDM4E (0.43) ALDH1A1KDM4EMAPTGAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 192 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250319060-A1 METHODS FOR THE PROPHYLAXIS AND TREATMENT OF COVID AND COVID-19 TRAN LLOYD HUNG LOI (US) 2025-10-16 US claimed
EP-4594325-A1 PEG-MODIFIED CYCLIC DIPEPTIDES Novmetapharma Co., Ltd. (KR) 2025-08-06 EP claimed
WO-2025088052-A1 CYCLIC ANALOGUE OF GLYCINE-PROLINE FOR USE IN THE PREVENTION AND/OR TREATMENT OF MEDICAL IMPLANT-RELATED FIBROSIS ROUSSELOT BV (BE) 2025-05-01 WO claimed
CN-119770491-A Application of cycloglycine-proline in preparing medicine for treating binge eating disease 北京大学 2025-04-08 CN claimed
CN-119775430-A Mineral composite peptide and preparation and application thereof 中国科学院烟台海岸带研究所 2025-04-08 CN claimed
US-20250049883-A1 ANIMAL, FUNGAL AND MARINE SOURCES OF CGP AND INCREASED CGP CONCENTRATION FOR DISEASE MANAGEMENT AND FOR TREATMENT OF NON-NEUROLOGICAL AND/OR NEUROLOGICAL CONDITIONS THE CGP LAB LTD (NZ) 2025-02-13 US claimed
US-12216119-B2 IGF-1 analysis, adjustment and disease management of non-neurological and/or neurological conditions THE CGP LAB LIMITED (NZ) 2025-02-04 US claimed
EP-4452270-A1 ANIMAL, FUNGAL AND MARINE SOURCES OF CGP AND INCREASED CGP CONCENTRATION FOR DISEASE MANAGEMENT AND FOR TREATMENT OF NON-NEUROLOGICAL AND/OR NEUROLOGICAL CONDITIONS THE CGP LAB LIMITED (NZ) 2024-10-30 EP claimed
CN-118613263-A CGP of animal, fungal and marine biological origin and increased cGP concentrations for disease management and treatment of non-neurological and/or neurological disorders CGP实验室有限公司 2024-09-06 CN claimed
US-20240140955-A1 PEG-MODIFIED CYCLIC DIPEPTIDES NOVMETAPHARMA CO., LTD. (KR) 2024-05-02 US claimed
WO-2024069524-A1 PEG-MODIFIED CYCLIC DIPEPTIDES NOVMETAPHARMA CO., LTD. (KR) 2024-04-04 WO claimed
US-20230218596-A1 METHODS INVOLVING NEUTROPHIL ELASTASE INHIBITOR ALVELESTAT FOR TREATING CORONAVIRUS INFECTION MEREO BIOPHARMA 4 LIMITED (GB) 2023-07-13 US claimed
WO-2023113623-A1 ANIMAL, FUNGAL AND MARINE SOURCES OF CGP AND INCREASED CGP CONCENTRATION FOR DISEASE MANAGEMENT AND FOR TREATMENT OF NON-NEUROLOGICAL AND/OR NEUROLOGICAL CONDITIONS THE CGP LAB LIMITED (NZ) 2023-06-22 WO claimed
EP-4138906-A1 METHODS FOR THE PROPHYLAXIS AND TREATMENT OF COVID AND COVID-19 Tran, Lloyd Hung Loi (US) 2023-03-01 EP claimed
EP-4743102-A1 COLLAGEN PEPTIDE COMPOSITION AND USE THEREOF IN AMELIORATING NEUROLOGICAL CONDITIONS AND FIBROSIS Rousselot BV (BE) 2026-05-20 EP disclosed
EP-4714452-A1 METHODS FOR TREATING SARS COV-2 INFECTIONS Gilead Sciences, Inc. (US) 2026-03-25 EP disclosed
EP-4702027-A1 4-AMINOPYRROLO[2,1-F][1,2,4]TRIAZINE C-NUCLEOSIDE COMPOUNDS AND METHODS FOR TREATMENT OF VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2026-03-04 EP disclosed
EP-1513842-A1 SUBSTITUTED HEXAHYDROPYRROLO (1,2-A)PYRAZINES, OCTAHYDROPYRIDO(1,2-A)PYRAZINES AND DECAHYDROPYRAZINO(1,2-A)AZEPINES NOVO NORDISK A/S (DK) 2005-03-16 EP disclosed
US-20040023946-A1 Substituted hexahydropyrrolo[1,2-a]pyrazines, octahydropyrido[1,2-a]-pyrazines and decahydropyrazino[1,2-a]azepines VTVX HOLDINGS II LLC 2004-02-05 US disclosed
WO-2003104235-A1 SUBSTITUTED HEXAHYDROPYRROLO[1,2-A]PYRAZINES, OCTAHYDROPYRIDO[1,2-A]PYRAZINES AND DECAHYDROPYRAZINO[1,2-A]AZEPINES NOVO NORDISK A/S (DK) 2003-12-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040023946-A1 Substituted hexahydropyrrolo[1,2-a]pyrazines, octahydropyrido[1,2-a]-pyrazines and decahydropyrazino[1,2-a]azepines HRH2, HRH4, HRH1 ALDH1A1 835/4885KDM4E 1409/4885MAPT 1954/4885
US-20240140955-A1 PEG-MODIFIED CYCLIC DIPEPTIDES LNPEP, ANPEP, DNPEP ALDH1A1 1719/4885KDM4E 2288/4885MAPT 3200/4885
US-20250319060-A1 METHODS FOR THE PROPHYLAXIS AND TREATMENT OF COVID AND COVID-19 ACE, ACE2, LPO ALDH1A1 1640/4885KDM4E 1900/4885MAPT 1277/4885
US-20230218596-A1 METHODS INVOLVING NEUTROPHIL ELASTASE INHIBITOR ALVELESTAT FOR TREATING CORONAVIRUS INFECTION SERPINB1, ELANE, MPO ALDH1A1 3704/4885KDM4E 4221/4885MAPT 2208/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.