Solriamfetol

Solriamfetol

SCHEMBL42525

NC(=O)OC[C@@H](N)Cc1ccccc1

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.56
CYP1A2 P05177 1/20 0.56
CYP2D6 P10635 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
EPHX1 P07099 2/20 0.55
MMP2 P08253 4/20 0.53
ALPI P09923 1/20 0.52
PTGS1 P23219 1/20 0.52
XIAP P98170 1/20 0.52
SLC7A5 Q01650 1/20 0.52
LMNA P02545 1/20 0.50
SCN4A P35499 2/20 0.49
ANPEP P15144 1/20 0.48
SRR Q9GZT4 2/20 0.47
SLC1A3 P43003 1/20 0.47
SLC1A2 P43004 1/20 0.47
SLC1A1 P43005 1/20 0.47
TACR1 P25103 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Solriamfetol SCHEMBL42526 1.00 PKM (0.56) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL2739637 1.00 PKM (0.56) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL30929348 1.00 PKM (0.56) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL30929349 1.00 PKM (0.56) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL8430382 0.98 PKM (0.54) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL28413501 0.98 PKM (0.54) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL4987496 0.98 PKM (0.54) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL8426383 0.98 PKM (0.54) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL30518836 0.97 PKM (0.53) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL30518840 0.95 PKM (0.51) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 211 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240239740-A1 TREATMENT OF SLEEP-WAKE DISORDERS SK BIOPHARMACEUTICALS CO LTD (KR) 2024-07-18 US claimed
US-20230278950-A1 METHODS FOR TREATING ATTENTION-DEFICIT/HYPERACTIVITY DISORDER SK BIOPHARMACEUTICALS CO LTD (KR) 2023-09-07 US claimed
US-11524935-B2 Methods for treating attention-deficit/hyperactivity disorder SK BIOPHARMACEUTICALS CO., LTD. (KR) 2022-12-13 US claimed
US-20210078943-A1 TREATMENT OF SLEEP-WAKE DISORDERS SK BIOPHARMACEUTICALS CO LTD (KR) 2021-03-18 US claimed
US-20210070694-A1 METHODS FOR TREATING ATTENTION-DEFICIT/HYPERACTIVITY DISORDER SK BIOPHARMACEUTICALS CO LTD (KR) 2021-03-11 US claimed
EP-3552604-B1 COMPOSITIONS FOR TREATING DRUG ADDICTION AND IMPROVING ADDICTION-RELATED BEHAVIOR SK BIOPHARMACEUTICALS CO LTD (KR) 2020-12-16 EP claimed
EP-3552604-A1 COMPOSITIONS FOR TREATING DRUG ADDICTION AND IMPROVING ADDICTION-RELATED BEHAVIOR SK Biopharmaceuticals Co., Ltd. (KR) 2019-10-16 EP claimed
US-20190194125-A1 METHODS FOR TREATING ATTENTION-DEFICIT/HYPERACTIVITY DISORDER SK BIOPHARMACEUTICALS CO LTD (KR) 2019-06-27 US claimed
EP-3308785-A2 USE OF FLECAINIDE AS AN ANTI-CONNEXIN AGENT AND METHOD FOR POTENTIATING THE EFFECTS OF A PSYCHOTROPIC DRUG Commissariat à l'Energie Atomique et aux Energies Alternatives (FR) 2018-04-18 EP claimed
US-20170355668-A1 METHODS FOR TREATING ATTENTION-DEFICIT/HYPERACTIVITY DISORDER SK BIOPHARMACEUTICALS CO LTD (KR) 2017-12-14 US claimed
EP-1890684-A1 TREATMENT OF SLEEP-WAKE DISORDERS SK Holdings Co., Ltd. (KR) 2008-02-27 EP claimed
WO-2006133393-A1 TREATMENT OF SLEEP-WAKE DISORDERS SK HOLDINGS CO., LTD. (KR) 2006-12-14 WO claimed
EP-0873308-B1 O-CARBAMOYL-PHENYLALANINOL COMPOUNDS AND THEIR PHARMACEUTICALLY USEFUL SALTS SK CORP (KR) 2002-01-02 EP claimed
EP-0820438-B1 O-CARBAMOYL-PHENYLALANINOL HAVING SUBSTITUENT AT BENZENE RING, ITS PHARMACEUTICALLY USEFUL SALTS AND METHOD FOR PREPARING THE SAME SK CORP (KR) 2001-06-20 EP claimed
US-6140532-A O-carbamoyl-phenylalaninol having substituent at benzene ring, its pharmaceutically useful salts and method for preparing the same SK CORPORATION (US) 2000-10-31 US claimed
EP-0873308-A1 O-CARBAMOYL-PHENYLALANINOL COMPOUNDS, THEIR PHARMACEUTICALLY USEFUL SALTS AND PROCESS FOR PREPARING THE SAME SK Corporation (KR) 1998-10-28 EP claimed
US-5756817-A TREATMENT OF DISEASES OF CENTRAL NERVOUS SYSTEMS YUKONG LIMITED (KR) 1998-05-26 US claimed
WO-1998015526-A1 O-CARBAMOYL-PHENYLALANINOL COMPOUNDS, THEIR PHARMACEUTICALLY USEFUL SALTS AND PROCESS FOR PREPARING THE SAME SK CORPORATION (KR) 1998-04-16 WO claimed
EP-0820438-A1 O-CARBAMOYL-PHENYLALANINOL HAVING SUBSTITUENT AT BENZENE RING, ITS PHARMACEUTICALLY USEFUL SALTS AND METHOD FOR PREPARING THE SAME YUKONG LIMITED (KR) 1998-01-28 EP claimed
WO-1996032375-A1 O-CARBAMOYL-PHENYLALANINOL HAVING SUBSTITUENT AT BENZENE RING, ITS PHARMACEUTICALLY USEFUL SALTS AND METHOD FOR PREPARING THE SAME YUKONG LIMITED (KR) 1996-10-17 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210070694-A1 METHODS FOR TREATING ATTENTION-DEFICIT/HYPERACTIVITY DISORDER CHAT, SLC6A3, SLC6A2 PKM 3986/4885CYP1A2 1712/4885CYP2D6 1271/4885
US-11524935-B2 Methods for treating attention-deficit/hyperactivity disorder CHAT, SLC6A3, SLC6A2 PKM 3986/4885CYP1A2 1712/4885CYP2D6 1271/4885
US-20230278950-A1 METHODS FOR TREATING ATTENTION-DEFICIT/HYPERACTIVITY DISORDER CHAT, SLC6A3, SLC6A2 PKM 3986/4885CYP1A2 1712/4885CYP2D6 1271/4885
US-20240239740-A1 TREATMENT OF SLEEP-WAKE DISORDERS HCRTR1, HCRTR2, MTNR1B PKM 3390/4885CYP1A2 119/4885CYP2D6 264/4885
US-20210078943-A1 TREATMENT OF SLEEP-WAKE DISORDERS HCRTR1, HCRTR2, MTNR1B PKM 3390/4885CYP1A2 119/4885CYP2D6 264/4885
US-20170355668-A1 METHODS FOR TREATING ATTENTION-DEFICIT/HYPERACTIVITY DISORDER CHAT, SLC6A3, SLC6A2 PKM 3986/4885CYP1A2 1712/4885CYP2D6 1271/4885
US-20190194125-A1 METHODS FOR TREATING ATTENTION-DEFICIT/HYPERACTIVITY DISORDER CHAT, SLC6A3, SLC6A2 PKM 3986/4885CYP1A2 1712/4885CYP2D6 1271/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.