Solriamfetol

Solriamfetol

SCHEMBL8430382

Cl.NC(=O)OC[C@H](N)Cc1ccccc1

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Solriamfetol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS1 known ✓ P23219 1/20 0.50
SCN4A known ✓ P35499 2/20 0.47
TACR1 known ✓ P25103 1/20 0.45
PKM P14618 2/20 0.54
CYP1A2 P05177 1/20 0.54
CYP2D6 P10635 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
EPHX1 P07099 2/20 0.53
MMP2 P08253 3/20 0.51
ALPI P09923 1/20 0.50
XIAP P98170 1/20 0.50
SLC7A5 Q01650 1/20 0.50
SRR Q9GZT4 2/20 0.49
LMNA P02545 1/20 0.49
ANPEP P15144 1/20 0.47
SLC1A3 P43003 1/20 0.46
SLC1A2 P43004 1/20 0.46
SLC1A1 P43005 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Solriamfetol SCHEMBL4987496 1.00 PKM (0.54) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL28413501 1.00 PKM (0.54) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL8426383 1.00 PKM (0.54) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL42526 0.98 PKM (0.56) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL30929348 0.98 PKM (0.56) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL30929349 0.98 PKM (0.56) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL2739637 0.98 PKM (0.56) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL42525 0.98 PKM (0.56) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL30518836 0.95 PKM (0.53) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1
Solriamfetol SCHEMBL30518840 0.93 PKM (0.51) PKMCYP1A2CYP2D6SMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 148 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250352476-A1 FORMULATIONS OF (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE AXSOME MALTA LTD (MT) 2025-11-20 US claimed
US-20250340509-A1 COMPOSITIONS COMPRISING (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE AND USES THEREOF AXSOME MALTA LTD (MT) 2025-11-06 US claimed
US-12390419-B2 Formulations of (R)-2-amino-3-phenylpropyl carbamate AXSOME MALTA LTD. (MT) 2025-08-19 US claimed
US-12384743-B2 Compositions comprising (R)-2-amino-3-phenylpropyl carbamate and uses thereof AXSOME MALTA LTD. (MT) 2025-08-12 US claimed
WO-2025092882-A1 COMBINATION OF A NORADRENERGIC α2A RECEPTOR AGONIST AND A NOREPINEPHRINE DOPAMINE REUPTAKE INHIBITOR AND USE THEREOF IGNIS THERAPEUTICS (SUZHOU) LIMITED (CN) 2025-05-08 WO claimed
US-20240285538-A1 FORMULATIONS OF (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE WILMINGTON TRUST, NATIONAL ASSOCIATION 2024-08-29 US claimed
US-20240282425-A1 AUTHENTICATION METHODS AND SYSTEMS FOR DISPENSED PRESCRIPTIONS LOW GORDON KEITH (US) 2024-08-22 US claimed
US-11998639-B2 Formulations of (R)-2-amino-3-phenylpropyl carbamate AXSOME MALTA LTD. (MT) 2024-06-04 US claimed
EP-4364794-A2 SOLVATE FORM OF (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE Axsome Malta Ltd. (MT) 2024-05-08 EP claimed
EP-3509582-B1 SOLVATE FORM OF (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE AXSOME MALTA LTD (MT) 2023-12-20 EP claimed
US-20210205227-A1 FORMULATIONS OF (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE WILMINGTON TRUST, NATIONAL ASSOCIATION 2021-07-08 US claimed
US-20210053912-A1 Compositions comprising (R)-2-amino-3-phenylpropyl carbamate and uses thereof WILMINGTON TRUST, NATIONAL ASSOCIATION 2021-02-25 US claimed
US-10829443-B2 Solvate form of (R)-2-amino-3-phenylpropyl carbamate JAZZ PHARMACEUTICALS IRELAND LIMITED (IE) 2020-11-10 US claimed
US-20200085748-A1 FORMULATIONS OF (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE AXSOME MALTA LTD. (MT) 2020-03-19 US claimed
EP-3509581-A1 FORMULATIONS OF (R Jazz Pharmaceuticals International III Limited (BM) 2019-07-17 EP claimed
US-20190194126-A1 Solvate Form of (R)-2-amino-3-phenylpropyl carbamate WILMINGTON TRUST, NATIONAL ASSOCIATION 2019-06-27 US claimed
US-20190117578-A1 FORMULATIONS OF (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE WILMINGTON TRUST, NATIONAL ASSOCIATION 2019-04-25 US claimed
US-10195151-B2 Formulations of (R)-2-amino-3-phenylpropyl carbamate JAZZ PHARMACEUTICALS INTERNATIONAL III LIMITED (BM) 2019-02-05 US claimed
WO-2018048862-A1 FORMULATIONS OF ( R)-2-AMINO-3-PHENYLPROPYL CARBAMATE JAZZ PHARMACEUTICALS INTERNATIONAL III LIMITED (BM) 2018-03-15 WO claimed
US-20180064652-A1 FORMULATIONS OF (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE WILMINGTON TRUST, NATIONAL ASSOCIATION 2018-03-08 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (14 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240285538-A1 FORMULATIONS OF (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE PRCP, GRPR, CPS1 PTGS1 1208/4885SCN4A 2296/4885TACR1 34/4885
US-12390419-B2 Formulations of (R)-2-amino-3-phenylpropyl carbamate PRCP, GRPR, CPS1 PTGS1 1208/4885SCN4A 2296/4885TACR1 34/4885
US-20250340509-A1 COMPOSITIONS COMPRISING (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE AND USES THEREOF APC, PKD1, PKD2 PTGS1 3895/4885SCN4A 1149/4885TACR1 1239/4885
US-20250352476-A1 FORMULATIONS OF (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE CPS1, PRCP, GLS2 PTGS1 2197/4885SCN4A 1361/4885TACR1 66/4885
US-20180064652-A1 FORMULATIONS OF (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE PRCP, GRPR, CPS1 PTGS1 1208/4885SCN4A 2296/4885TACR1 34/4885
US-20210205227-A1 FORMULATIONS OF (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE PRCP, GRPR, CPS1 PTGS1 1208/4885SCN4A 2296/4885TACR1 34/4885
US-12384743-B2 Compositions comprising (R)-2-amino-3-phenylpropyl carbamate and uses thereof APC, PKD1, PKD2 PTGS1 3895/4885SCN4A 1149/4885TACR1 1239/4885
US-10829443-B2 Solvate form of (R)-2-amino-3-phenylpropyl carbamate APC, PKD1, PKD2 PTGS1 4001/4885SCN4A 1282/4885TACR1 795/4885
US-10195151-B2 Formulations of (R)-2-amino-3-phenylpropyl carbamate PRCP, GRPR, CPS1 PTGS1 1208/4885SCN4A 2296/4885TACR1 34/4885
US-20210053912-A1 Compositions comprising (R)-2-amino-3-phenylpropyl carbamate and uses thereof APC, PKD1, PKD2 PTGS1 3895/4885SCN4A 1149/4885TACR1 1239/4885
US-20190194126-A1 Solvate Form of (R)-2-amino-3-phenylpropyl carbamate APC, PKD1, PKD2 PTGS1 4001/4885SCN4A 1282/4885TACR1 795/4885
US-20190117578-A1 FORMULATIONS OF (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE PRCP, GRPR, CPS1 PTGS1 1208/4885SCN4A 2296/4885TACR1 34/4885
US-20200085748-A1 FORMULATIONS OF (R)-2-AMINO-3-PHENYLPROPYL CARBAMATE PRCP, GRPR, CPS1 PTGS1 1208/4885SCN4A 2296/4885TACR1 34/4885
US-11998639-B2 Formulations of (R)-2-amino-3-phenylpropyl carbamate PRCP, GRPR, CPS1 PTGS1 1208/4885SCN4A 2296/4885TACR1 34/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.