SCHEMBL4255735

SCHEMBL4255735

O=C1NC(=O)C2(N1)C(=O)N(Cc1ccccc1)c1ccc(Cl)cc12

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.52
MAPT P10636 3/20 0.52
AKR1A1 P14550 2/20 0.51
AKR1B1 P15121 2/20 0.51
PTGDR2 Q9Y5Y4 9/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CNR1 P21554 1/20 0.48
ALDH1A1 P00352 1/20 0.46
ALDH2 P05091 1/20 0.46
ALDH3A1 P30838 1/20 0.46
SCN9A Q15858 1/20 0.44
C5AR1 P21730 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4164476 0.90 CNR1 (0.51) TP53MAPTAKR1A1AKR1B1PTGDR2
SCHEMBL10960512 0.87 AKR1A1 (0.47) TP53MAPTAKR1A1AKR1B1PTGDR2
SCHEMBL11045654 0.87 TP53 (0.54) TP53MAPTAKR1A1AKR1B1CNR1
SCHEMBL4259885 0.87 ADAMTS5 (0.52) TP53MAPTSMN1; SMN2CNR1ALDH1A1
SCHEMBL4260419 0.87 PARK7 (0.51) AKR1A1AKR1B1PTGDR2CNR1ALDH1A1
SCHEMBL4254336 0.86 ALDH1A1 (0.51) TP53MAPTCNR1ALDH1A1SCN9A
SCHEMBL4167863 0.84 AKR1B1 (0.44) TP53MAPTAKR1A1AKR1B1PTGDR2
SCHEMBL4258971 0.83 TP53 (0.45) TP53MAPTAKR1A1AKR1B1PTGDR2
SCHEMBL2686520 0.83 PTGDR2 (0.63) AKR1A1AKR1B1PTGDR2
SCHEMBL4166000 0.82 HPGD (0.46) MAPTAKR1A1AKR1B1PTGDR2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090176851-A1 Use of Spiro [Imidazolidine-4, 3' -Indole] 2, 2', 5' (1H) Triones for Treatment of Conditions Associated with Vanilloid Receptor 1 ASTRAZENECA AB (SE) 2009-07-09 US claimed
US-20090176851-A1 Use of Spiro [Imidazolidine-4, 3' -Indole] 2, 2', 5' (1H) Triones for Treatment of Conditions Associated with Vanilloid Receptor 1 ASTRAZENECA AB (SE) 2009-07-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090176851-A1 Use of Spiro [Imidazolidine-4, 3' -Indole] 2, 2', 5' (1H) Triones for Treatment of Conditions Associated with Vanilloid Receptor 1 TRPV1, TRPV2, TRPV3 TP53 3194/4885MAPT 3349/4885AKR1A1 317/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.