SCHEMBL4285889

SCHEMBL4285889

Cn1nc(C(C)(C)C)cc1N(Cc1cccc(N2CCOCC2)c1)CC1CCCCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGXT P21549 1/20 0.38
HTR2C P28335 3/20 0.37
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
HTR1A P08908 2/20 0.35
HTR1D P28221 1/20 0.35
HTR1B P28222 1/20 0.35
PRKDC P78527 3/20 0.35
MAPK14 Q16539 2/20 0.34
ATM Q13315 4/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
PIK3C3 Q8NEB9 2/20 0.33
AKT1 P31749 1/20 0.33
PIK3CA P42336 1/20 0.33
AOC3 Q16853 1/20 0.33
CCKBR P32239 1/20 0.33
HTR2A P28223 2/20 0.33
HTR7 P34969 2/20 0.33
CTSL P07711 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4282621 0.90 AGXT (0.36) AGXTHTR2CHCRTR1HCRTR2HTR1A
SCHEMBL4287197 0.85 AGXT (0.37) AGXTHTR2CHCRTR1HCRTR2HTR1A
SCHEMBL5141171 0.83 AGXT (0.40) AGXTHCRTR1HCRTR2HTR1AHTR1D
SCHEMBL5141914 0.82 AGXT (0.39) AGXTHCRTR1HCRTR2HTR1AHTR1D
SCHEMBL4128842 0.76 KDM4E (0.35) AGXTHTR2CHCRTR1HCRTR2HTR1A
SCHEMBL4133677 0.72 TPH1 (0.33) AGXTHTR2CHCRTR1HCRTR2PRKDC
SCHEMBL4128912 0.70 PDE5A (0.41) MEN1KMT2A
SCHEMBL4142910 0.67 HSP90AA1 (0.37) AGXTHTR1AHTR1DHTR1BPRKDC
SCHEMBL4282837 0.67 HTR7 (0.40) AGXTMEN1KMT2AHTR7
SCHEMBL8042201 0.66 AGXT (0.50) AGXTHCRTR1HCRTR2AOC3PRMT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071706-A1 PYRAZOLEPYRIMIDINE COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2009-06-11 WO disclosed