SCHEMBL4294715

SCHEMBL4294715

[2H]C([2H])([2H])c1cc(OC)cc(C([2H])([2H])[2H])c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
ACHE P22303 2/20 0.42
CYP1A1 P04798 5/20 0.40
CYP1B1 Q16678 5/20 0.40
CYP3A4 P08684 5/20 0.39
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA12 O43570 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
TDP1 Q9NUW8 2/20 0.36
MAPK1 P28482 1/20 0.36
CYP1A2 P05177 3/20 0.36
CYP2E1 P05181 2/20 0.36
CYP2C8 P10632 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2A6 P11509 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP4B1 P13584 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16707188 0.95 ALDH1A1 (0.48) ALDH1A1ACHECYP1A1CYP1B1CYP3A4
SCHEMBL145855 0.79 ALDH1A1 (0.62) ALDH1A1ACHECYP1A1CYP1B1CYP3A4
SCHEMBL29587173 0.77 ALDH1A1 (0.59) ALDH1A1ACHECYP1A1CYP1B1CYP3A4
SCHEMBL12501 0.73 ALDH1A1 (0.73) ALDH1A1ACHECYP1A1CYP1B1CYP3A4
SCHEMBL16116743 0.72 ALDH1A1 (0.42) ALDH1A1ACHECYP3A4TDP1MAPK1
SCHEMBL16550555 0.72
1,3,5-Trimethoxybenzene SCHEMBL28493 0.71 ALDH1A1 (1.00) ALDH1A1CYP1A1CYP1B1CYP3A4CA1
1,3,5-Trimethoxybenzene SCHEMBL31747526 0.71 ALDH1A1 (0.69) ALDH1A1CYP1A1CYP1B1CYP3A4CA1
1,3,5-Trimethoxybenzene SCHEMBL31747507 0.71 ALDH1A1 (0.69) ALDH1A1CYP1A1CYP1B1CYP3A4CA1
SCHEMBL4342018 0.70 ALDH1A1 (0.50) ALDH1A1ACHECYP1A1CYP1B1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9770432-B2 Deuterated benzopyran compounds and the use in the treatment of pain and inflammation GUANGZHOU INSTITUTES OF BIOMEDICINE AND HEALTH, CHINESE ACADEMY OF SCIENCES (CN) 2017-09-26 US disclosed
US-9763914-B2 Deuterated benzopyran compounds and application thereof GUANGZHOU INSTITUTES OF BIOMEDICINE AND HEALTH, CHINESE ACADEMY OF SCIENCES (CN) 2017-09-19 US disclosed
US-20170020843-A1 DEUTERATED BENZOPYRAN COMPOUNDS AND APPLICATION THEREOF INFLAMAX PHARMACEUTICALS LIMITED (CN) 2017-01-26 US disclosed
US-20160287556-A1 DEUTERATED BENZOPYRAN COMPOUNDS AND APPLICATION THEREOF INFLAMAX PHARMACEUTICALS LIMITED (CN) 2016-10-06 US disclosed
EP-2845854-B1 DEUTERATED BENZOPYRAN COMPOUND AND APPLICATION THEREOF GUANGZHOU INST BIOMED & HEALTH (CN) 2016-09-21 EP disclosed
US-9371305-B2 Deuterated benzopyran compounds and application thereof GUANGZHOU INSTITUTES OF BIOMEDICINE AND HEALTH, CHINESE ACADEMY OF SCIENCES (CN) 2016-06-21 US disclosed
US-20150133538-A1 Deuterated Benzopyran Compounds and Application Thereof GUANGZHOU INSTITUTES OF BIOMEDICINE AND HEALTH, CHINESE ACADEMY OF SCIENCES (CN) 2015-05-14 US disclosed
EP-2845854-A1 DEUTERATED BENZOPYRAN COMPOUND AND APPLICATION THEREOF Guangzhou Institute Of Biomedicine And Health, Chinese Academy Of Sciences (CN) 2015-03-11 EP disclosed
CN-102757417-B Deuterated benzopyran compound and application thereof GUANGZHOU INST BIOMED & HEALTH 2014-09-24 CN disclosed
CN-102757417-A Deuterated benzopyran compound and application thereof GUANGZHOU INST BIOMED & HEALTH 2012-10-31 CN disclosed
US-20090270469-A1 SUBSTITUTED OXAZOLIDINONES AUSPEX PHARMACEUTICALS, INC. (US) 2009-10-29 US disclosed
US-20090270469-A1 SUBSTITUTED OXAZOLIDINONES AUSPEX PHARMACEUTICALS, INC. (US) 2009-10-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090270469-A1 SUBSTITUTED OXAZOLIDINONES MUSK, MYLK2, PYGM ALDH1A1 2157/4885ACHE 405/4885CYP1A1 2250/4885
US-20150133538-A1 Deuterated Benzopyran Compounds and Application Thereof PTGS2, HPGDS, PTGS1 ALDH1A1 324/4885ACHE 2101/4885CYP1A1 113/4885
US-20160287556-A1 DEUTERATED BENZOPYRAN COMPOUNDS AND APPLICATION THEREOF PTGS2, HPGDS, PTGS1 ALDH1A1 324/4885ACHE 2101/4885CYP1A1 113/4885
US-20170020843-A1 DEUTERATED BENZOPYRAN COMPOUNDS AND APPLICATION THEREOF PTGS2, HPGDS, PTGS1 ALDH1A1 324/4885ACHE 2101/4885CYP1A1 113/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.