SCHEMBL4314169

SCHEMBL4314169

Cc1c(C2=CCC(c3ccccc3)([As](C)C)CC2)n(CC(O)CN(C)C)c2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DNM1 Q05193 5/20 0.47
KDM4E B2RXH2 5/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CRY1 Q16526 6/20 0.39
CRY2 Q49AN0 6/20 0.39
PER2 O15055 5/20 0.39
ALDH1A1 P00352 3/20 0.39
MYLK Q15746 2/20 0.38
LMNA P02545 2/20 0.37
ALOX15 P16050 2/20 0.37
HSD17B10 Q99714 1/20 0.37
MAPT P10636 2/20 0.37
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
TSHR P16473 1/20 0.36
NPY1R P25929 1/20 0.36
NPY2R P49146 1/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL734333 0.87 DNM1 (0.49) DNM1KDM4ESMN1; SMN2CRY1CRY2
SCHEMBL734385 0.69 DNM1 (0.55) DNM1KDM4ESMN1; SMN2CRY1CRY2
SCHEMBL734760 0.67 DHFR (0.40) LMNAMAPTL3MBTL1
SCHEMBL18862339 0.59 KDM4E (0.97) DNM1KDM4ESMN1; SMN2ALDH1A1LMNA
SCHEMBL735924 0.58 ALDH1A1 (0.44) DNM1KDM4ESMN1; SMN2CRY1CRY2
SCHEMBL15383951 0.57 PER2 (1.00) DNM1SMN1; SMN2CRY1CRY2PER2
SCHEMBL4878312 0.56 MYLK (0.73) DNM1SMN1; SMN2CRY1CRY2PER2
SCHEMBL20462136 0.56 PER2 (0.63) DNM1KDM4ECRY1CRY2PER2
SCHEMBL8113510 0.56 MYLK (1.00) DNM1MYLK
SCHEMBL21467809 0.55 DNM1 (0.71) DNM1SMN1; SMN2CRY1CRY2PER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044016-A2 4-HETEROARYL-SUBSTITUTED 1-AMINOCYCLOHEXANE-1-AND CYCLOHEXENE-1-DERIVATIVES HAVING EFFECTS ON THE OPIOD RECEPTOR SYSTEM Grünenthal GmbH (DE) 2009-04-08 EP claimed
WO-2008009415-A2 4-HETEROARYL-SUBSTITUTED 1-AMINOCYCLOHEXANE-1- AND CYCLOHEXENE-1-DERIVATIVES HAVING EFFECTS ON THE OPIOD RECEPTOR SYSTEM Grünenthal GmbH (DE) 2008-01-24 WO claimed