Known targets — ChEMBL curated mechanism
ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO
The experimentally established mechanism targets of Sulfamate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.
Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | MEN1 known ✓ | O00255 | 1/20 | 0.36 |
| ▸ | CA1 | P00915 | 6/20 | 0.80 |
| ▸ | CA2 | P00918 | 6/20 | 0.80 |
| ▸ | CA5A | P35218 | 3/20 | 0.80 |
| ▸ | CA5B | Q9Y2D0 | 3/20 | 0.80 |
| ▸ | CA9 | Q16790 | 3/20 | 0.80 |
| ▸ | CA7 | P43166 | 3/20 | 0.80 |
| ▸ | TSHR | P16473 | 3/20 | 0.80 |
| ▸ | CA4 | P22748 | 2/20 | 0.80 |
| ▸ | CA6 | P23280 | 2/20 | 0.80 |
| ▸ | NT5E | P21589 | 1/20 | 0.80 |
| ▸ | CA12 | O43570 | 1/20 | 0.40 |
| ▸ | TDP1 | Q9NUW8 | 1/20 | 0.39 |
| ▸ | BLM | P54132 | 3/20 | 0.38 |
| ▸ | KDM4E | B2RXH2 | 2/20 | 0.38 |
| ▸ | ALDH1A1 | P00352 | 1/20 | 0.36 |
| ▸ | KMT2A | Q03164 | 1/20 | 0.36 |
| ▸ | CYP2C19 | P33261 | 2/20 | 0.33 |
| ▸ | LMNA | P02545 | 1/20 | 0.33 |
| ▸ | SLC6A6 | P31641 | 1/20 | 0.33 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| Sulfamate SCHEMBL502342 | 1.00 | CA1 (0.80) | CA1CA2CA5ACA5BCA9 | |
| Sulfamate SCHEMBL11895110 | 1.00 | — | — | |
| Sulfamate SCHEMBL16041710 | 0.95 | CA1 (0.89) | CA1CA2CA5ACA5BCA9 | |
| Sulfamate SCHEMBL4614086 | 0.95 | — | — | |
| Sulfamate SCHEMBL2341482 | 0.95 | — | — | |
| Sulfamate SCHEMBL29826201 | 0.95 | — | — | |
| Sulfamate SCHEMBL42731 | 0.95 | — | — | |
| Sulfamate SCHEMBL5147247 | 0.95 | — | — | |
| Sulfamate SCHEMBL3702264 | 0.90 | — | — | |
| Sulfamate SCHEMBL15843606 | 0.90 | — | — |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| CN-118792715-A | Super-hydrophilic nano-coating diamond wire saw and manufacturing method thereof | 镇江原轼新型材料有限公司 | 2024-10-18 | — | — | CN | claimed |
| CN-117601291-A | Wire saw and manufacturing method thereof | 镇江原轼新型材料有限公司 | 2024-02-27 | — | — | CN | claimed |
| CN-118792715-A | Super-hydrophilic nano-coating diamond wire saw and manufacturing method thereof | 镇江原轼新型材料有限公司 | 2024-10-18 | — | — | CN | disclosed |
| CN-117601291-A | Wire saw and manufacturing method thereof | 镇江原轼新型材料有限公司 | 2024-02-27 | — | — | CN | disclosed |
| CN-117601290-A | Wire saw and method for manufacturing wire saw | 镇江原轼新型材料有限公司 | 2024-02-27 | — | — | CN | disclosed |
| US-11810691-B2 | Aluminum base wire | SUMITOMO ELECTRIC INDUSTRIES, LTD. (JP) | 2023-11-07 | — | — | US | disclosed |
| CN-113544315-B | Aluminum-based wire rod | 住友电气工业株式会社 | 2023-09-29 | — | — | CN | disclosed |
| US-20220139593-A1 | ALUMINUM BASE WIRE | SUMITOMO ELECTRIC INDUSTRIES, LTD. (JP) | 2022-05-05 | — | — | US | disclosed |
| CN-113544315-A | Aluminum-based wire rod | 住友电气工业株式会社 | 2021-10-22 | — | — | CN | disclosed |
| US-9263162-B2 | Method for manufacturing microstructure | CANON KABUSHIKI KAISHA (JP) | 2016-02-16 | — | — | US | disclosed |
| US-9040227-B2 | Microstructure manufacturing method | CANON KABUSHIKI KAISHA (JP) | 2015-05-26 | — | — | US | disclosed |
| US-20150060405-A1 | METHOD FOR MANUFACTURING MICROSTRUCTURE | CANON KABUSHIKI KAISHA (JP) | 2015-03-05 | — | — | US | disclosed |
| US-20130118793-A1 | METHOD FOR FILLING THROUGH HOLE OF SUBSTRATE WITH METAL AND SUBSTRATE | CANON KABUSHIKI KAISHA (JP) | 2013-05-16 | — | — | US | disclosed |
| US-20120219916-A1 | MICROSTRUCTURE MANUFACTURING METHOD | CANON KABUSHIKI KAISHA (JP) | 2012-08-30 | — | — | US | disclosed |
| WO-2012011230-A1 | METHOD FOR FILLING THROUGH HOLE OF SUBSTRATE WITH METAL AND SUBSTRATE | CANON KABUSHIKI KAISHA (JP) | 2012-01-26 | — | — | WO | disclosed |
| US-20060177609-A1 | Ink-jet recording sheet | KONICA MINOLTA HOLDINGS, INC. (JP) | 2006-08-10 | — | — | US | disclosed |
| US-20040185194-A1 | comprises ink receptive layer containing silica microparticles (formed by pulverization of silica powder) and water-soluble resin; improved gloss | KONICA MINOLTA HOLDINGS, INC. (JP) | 2004-09-23 | — | — | US | disclosed |
| US-6278764-B1 | High efficiency replicated x-ray optics and fabrication method | THE REGENTS OF THE UNVIERSITY OF CALIFORNIA | 2001-08-21 | — | — | US | disclosed |
| WO-2001008162-A1 | HIGH EFFICIENCY REPLICATED X-RAY OPTICS AND FABRICATION METHOD | THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) | 2001-02-01 | — | — | WO | disclosed |
| US-4785137-A | HERMETIC SEALED CONTAINER | ALLIED CORPORATION (US) | 1988-11-15 | — | — | US | disclosed |