SCHEMBL4329797

SCHEMBL4329797

N=C(N)Nc1nc(-c2ccc(OC(=O)c3ccc(-c4ccccc4)cc3)cc2)cs1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.56
NPC1 O15118 3/20 0.54
RAB9A P51151 3/20 0.54
MAPT P10636 3/20 0.54
PKM P14618 1/20 0.54
SCD O00767 1/20 0.52
CASP3 P42574 1/20 0.52
SENP7 Q9BQF6 1/20 0.52
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
CSNK2A1 P68400 1/20 0.50
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
PARP1 P09874 1/20 0.49
PHGDH O43175 2/20 0.48
APP P05067 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4331871 0.90 ADORA3 (0.58) ADORA3NPC1RAB9AMAPTCASP3
SCHEMBL4333461 0.89 RAB9A (0.53) ADORA3NPC1RAB9AMAPTPKM
SCHEMBL4322683 0.88 MEN1 (0.60) ADORA3NPC1RAB9AMAPTPKM
SCHEMBL4330728 0.86 ADORA3 (0.48) ADORA3NPC1RAB9AMAPTPKM
SCHEMBL4324209 0.85 RAB9A (0.44) ADORA3NPC1RAB9AMAPTPKM
SCHEMBL3598628 0.85 MAPT (0.58) ADORA3NPC1RAB9AMAPTSCD
SCHEMBL4326708 0.83 MAPT (0.53) ADORA3NPC1RAB9AMAPTPKM
SCHEMBL4342353 0.83 RAB9A (0.50) ADORA3NPC1RAB9AMAPTPKM
SCHEMBL4330706 0.83 SCD (0.70) ADORA3NPC1RAB9AMAPTSCD
SCHEMBL3615150 0.83 MEN1 (0.55) ADORA3NPC1RAB9AMAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009146013-A1 MYOSIN LIGHT CHAIN PHOSPHATASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2009-12-03 WO claimed
WO-2009146013-A1 MYOSIN LIGHT CHAIN PHOSPHATASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2009-12-03 WO disclosed
WO-2009146013-A1 MYOSIN LIGHT CHAIN PHOSPHATASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2009-12-03 WO disclosed