SCHEMBL4333461

SCHEMBL4333461

N=C(N)Nc1nc(-c2ccc(OC(=O)c3ccc4ccccc4c3)cc2)cs1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.53
NPC1 O15118 3/20 0.53
CSNK2A1 P68400 3/20 0.51
TDP1 Q9NUW8 1/20 0.51
MAPT P10636 3/20 0.50
GSTO1 P78417 1/20 0.50
PKM P14618 1/20 0.50
MEN1 O00255 6/20 0.49
KMT2A Q03164 6/20 0.49
KDM4E B2RXH2 2/20 0.49
ADORA3 P0DMS8 1/20 0.49
ALDH1A1 P00352 2/20 0.45
GAA P10253 2/20 0.45
SCD O00767 1/20 0.45
PTGES O14684 1/20 0.44
HPGD P15428 1/20 0.44
VCP P55072 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4329797 0.89 ADORA3 (0.56) RAB9ANPC1CSNK2A1MAPTPKM
SCHEMBL4331871 0.84 ADORA3 (0.58) RAB9ANPC1CSNK2A1MAPTGSTO1
SCHEMBL13578656 0.84 MEN1 (0.59) RAB9ANPC1CSNK2A1TDP1MAPT
SCHEMBL4342353 0.83 RAB9A (0.50) RAB9ANPC1CSNK2A1MAPTPKM
SCHEMBL4322683 0.82 MEN1 (0.60) RAB9ANPC1CSNK2A1MAPTGSTO1
SCHEMBL4330728 0.82 ADORA3 (0.48) RAB9ANPC1CSNK2A1TDP1MAPT
SCHEMBL4328007 0.82 ALDH1A1 (0.59) RAB9ANPC1CSNK2A1TDP1MAPT
SCHEMBL3608900 0.82 RAB9A (0.67) RAB9ANPC1CSNK2A1MAPTGSTO1
SCHEMBL30660072 0.82 RAB9A (0.67) RAB9ANPC1CSNK2A1MAPTGSTO1
SCHEMBL4324209 0.82 RAB9A (0.44) RAB9ANPC1CSNK2A1MAPTGSTO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009146013-A1 MYOSIN LIGHT CHAIN PHOSPHATASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2009-12-03 WO claimed
WO-2009146013-A1 MYOSIN LIGHT CHAIN PHOSPHATASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2009-12-03 WO disclosed