SCHEMBL4322683

SCHEMBL4322683

COc1cccc(-c2ccc(C(=O)Oc3ccc(-c4csc(NC(=N)N)n4)cc3)cc2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.60
KMT2A Q03164 6/20 0.60
ALDH1A1 P00352 3/20 0.60
NPC1 O15118 4/20 0.58
RAB9A P51151 4/20 0.58
HPGD P15428 1/20 0.58
HTT P42858 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
HSD17B10 Q99714 1/20 0.58
CSNK2A1 P68400 2/20 0.55
ADORA3 P0DMS8 1/20 0.54
MAPT P10636 4/20 0.53
THRB P10828 1/20 0.53
PAX8 Q06710 1/20 0.50
ATP4A P20648 2/20 0.49
ATP4B P51164 2/20 0.49
CYP3A4 P08684 2/20 0.48
PRKACA P17612 1/20 0.48
ROCK1 Q13464 1/20 0.48
PKM P14618 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4331871 0.91 ADORA3 (0.58) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL4329797 0.88 ADORA3 (0.56) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL3613302 0.84 ALDH1A1 (0.72) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL4333461 0.82 RAB9A (0.53) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL4330728 0.82 ADORA3 (0.48) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL4322678 0.81 ATP4A (0.70) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL3615150 0.81 MEN1 (0.55) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL3595657 0.79 PTGS2 (0.66) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL4324209 0.79 RAB9A (0.44) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL4326708 0.79 MAPT (0.53) MEN1KMT2AALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009146013-A1 MYOSIN LIGHT CHAIN PHOSPHATASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2009-12-03 WO claimed
WO-2009146013-A1 MYOSIN LIGHT CHAIN PHOSPHATASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2009-12-03 WO disclosed