SCHEMBL4336015

SCHEMBL4336015

Cc1ccc(C(=O)NCCCCn2cc(-c3ccccc3)c3ccc(C(=O)O)cc32)c(O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
SMYD2 Q9NRG4 1/20 0.41
SCN9A Q15858 3/20 0.41
S1PR1 P21453 1/20 0.39
CPT2 P23786 1/20 0.39
CPT1A P50416 1/20 0.39
CPT1B Q92523 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4320012 0.89 LMNA (0.46) NPC1RAB9ASMYD2SCN9ACPT2
SCHEMBL4327173 0.89 SCN9A (0.39) PTGS2SMYD2SCN9AS1PR1CPT2
SCHEMBL4331918 0.83 BRD4 (0.44) SMYD2SCN9ACPT2CPT1ACPT1B
SCHEMBL4319190 0.82 SLC22A12 (0.43) SMYD2SCN9AS1PR1CPT2CPT1A
SCHEMBL4324558 0.82 NPC1 (0.48) NPC1RAB9ASMN1; SMN2SMYD2SCN9A
SCHEMBL4321178 0.82 LMNA (0.51) NPC1RAB9ALMNAHTTALDH1A1
SCHEMBL4326354 0.81 NAMPT (0.46) SMYD2SCN9ACPT2CPT1ACPT1B
SCHEMBL4336046 0.81 LMNA (0.46) NPC1RAB9ASMN1; SMN2SCN9ALMNA
SCHEMBL4324640 0.81 HCRTR1 (0.54) RAB9ASMN1; SMN2SCN9AKDM4EALDH1A1
SCHEMBL4333849 0.81 DRD2 (0.46) SMN1; SMN2SCN9ACPT2CPT1ACPT1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009147121-A1 CARBOXYL SUBSTITUTED INDOLES FOR USE AS PPAR ALPHA MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-10 WO claimed
WO-2009147121-A1 CARBOXYL SUBSTITUTED INDOLES FOR USE AS PPAR ALPHA MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-10 WO disclosed