SCHEMBL4324640

SCHEMBL4324640

CCOc1ccccc1C(=O)NCCCCn1cc(-c2ccccc2)c2ccc(C(=O)O)cc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.54
TSHR P16473 1/20 0.46
ALDH1A1 P00352 3/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HIF1A Q16665 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HTR7 P34969 2/20 0.42
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
CYP2C19 P33261 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4324512 0.93 MEN1 (0.52) HCRTR1TSHRALDH1A1HDAC3HDAC1
SCHEMBL4321178 0.84 LMNA (0.51) ALDH1A1MEN1KMT2AHPGDRAB9A
SCHEMBL4319190 0.83 SLC22A12 (0.43) HDAC1SCN9ACNR1CNR2
SCHEMBL4320012 0.82 LMNA (0.46) ALDH1A1L3MBTL1MEN1KMT2ANPSR1
SCHEMBL4335709 0.82 CYP2C19 (0.39) ALDH1A1CYP1A2CYP2C9CYP2C19SCN9A
SCHEMBL4331873 0.82 NPC1 (0.50) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL4336015 0.81 NPC1 (0.41) ALDH1A1KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL4336046 0.81 LMNA (0.46) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL4333849 0.81 DRD2 (0.46) MAPTSMN1; SMN2SCN9A
SCHEMBL4330789 0.80 NPC1 (0.49) HDAC3HPGDSMN1; SMN2RAB9ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009147121-A1 CARBOXYL SUBSTITUTED INDOLES FOR USE AS PPAR ALPHA MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-10 WO claimed
WO-2009147121-A1 CARBOXYL SUBSTITUTED INDOLES FOR USE AS PPAR ALPHA MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-10 WO disclosed