SCHEMBL4331918

SCHEMBL4331918

Cc1ccc(C(=O)NCCCCn2cc(-c3ccccc3)c3ccc(C(=O)O)cc32)c(Cl)n1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.44
SMYD2 Q9NRG4 1/20 0.40
EGFR P00533 1/20 0.40
PDE4A P27815 3/20 0.40
PDE4B Q07343 3/20 0.40
PDE4C Q08493 3/20 0.40
PDE4D Q08499 3/20 0.40
PPARG P37231 2/20 0.39
CNR1 P21554 1/20 0.39
SCN9A Q15858 1/20 0.39
SLC22A12 Q96S37 1/20 0.39
AGTR1 P30556 2/20 0.38
AGTR2 P50052 1/20 0.38
CPT2 P23786 1/20 0.37
CPT1A P50416 1/20 0.37
CPT1B Q92523 1/20 0.37
DHODH Q02127 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4336015 0.83 NPC1 (0.41) SMYD2PDE4APDE4BPDE4CPDE4D
SCHEMBL4320012 0.83 LMNA (0.46) SMYD2SCN9ASLC22A12CPT2CPT1A
SCHEMBL4333849 0.83 DRD2 (0.46) SCN9ACPT2CPT1ACPT1B
SCHEMBL4330789 0.81 NPC1 (0.49) PPARGSCN9ASLC22A12CPT2CPT1A
SCHEMBL4324558 0.80 NPC1 (0.48) SMYD2SCN9ASLC22A12CPT2CPT1A
SCHEMBL4321178 0.80 LMNA (0.51) PPARG
SCHEMBL4327173 0.80 SCN9A (0.39) SMYD2PPARGCNR1SCN9ACPT2
SCHEMBL4336046 0.79 LMNA (0.46) PPARGSCN9A
SCHEMBL4324640 0.79 HCRTR1 (0.54) CNR1SCN9A
SCHEMBL4335709 0.79 CYP2C19 (0.39) SMYD2PPARGCNR1SCN9ACPT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009147121-A1 CARBOXYL SUBSTITUTED INDOLES FOR USE AS PPAR ALPHA MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-10 WO claimed
WO-2009147121-A1 CARBOXYL SUBSTITUTED INDOLES FOR USE AS PPAR ALPHA MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-10 WO disclosed