SCHEMBL4339384

SCHEMBL4339384

COc1ccc(NC(=O)OCc2cc(CC(OC(C)C)C(=O)O)ccc2F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
FPR2 P25090 3/20 0.42
MAPT P10636 2/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 3/20 0.41
POLB P06746 2/20 0.41
SAE1 Q9UBE0 1/20 0.40
UBA2 Q9UBT2 1/20 0.40
PPARG P37231 2/20 0.40
PPARD Q03181 2/20 0.40
PPARA Q07869 2/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4341998 0.90 CYP1A2 (0.43) NPC1RAB9ASMN1; SMN2CYP1A2CYP2D6
SCHEMBL4348494 0.90 MGLL (0.40) NPC1RAB9ASMN1; SMN2CYP1A2CYP2D6
SCHEMBL4343670 0.89 TSHR (0.44) NPC1RAB9ASMN1; SMN2CYP1A2CYP2D6
SCHEMBL4333343 0.88 PPARA (0.44) SMN1; SMN2FPR2KMT2APPARGPPARD
SCHEMBL6652955 0.86 KDM4E (0.49) NPC1RAB9ASMN1; SMN2FPR2MAPT
SCHEMBL13810555 0.86 PPARG (0.41) NPC1RAB9ASMN1; SMN2CYP1A2CYP2D6
SCHEMBL4335156 0.86 NPC1 (0.50) NPC1RAB9ASMN1; SMN2CYP1A2CYP2D6
SCHEMBL4328737 0.84 FPR2 (0.48) NPC1RAB9ASMN1; SMN2CYP1A2CYP2D6
SCHEMBL4341155 0.84 ALDH1A1 (0.48) NPC1RAB9ASMN1; SMN2CYP1A2CYP2C9
SCHEMBL4337170 0.83 MMP1 (0.44) SMN1; SMN2CYP1A2CYP2D6CYP2C9HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7544835-B2 Carboxylic acid derivative and salt thereof EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-06-09 US disclosed
US-7544835-B2 Carboxylic acid derivative and salt thereof EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-06-09 US disclosed
US-7544835-B2 Carboxylic acid derivative and salt thereof EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-06-09 US disclosed