SCHEMBL434170

SCHEMBL434170

O=S(=O)(Cl)c1ccc(F)cc1Br

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.49
TRPV4 Q9HBA0 3/20 0.39
EPHX2 P34913 1/20 0.37
PTGES2 Q9H7Z7 6/20 0.36
PKM P14618 1/20 0.36
AKR1B1 P15121 2/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
CCR2 P41597 1/20 0.33
EPAS1 Q99814 1/20 0.33
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31645221 1.00 KMT2A (0.49) KMT2ATRPV4EPHX2PTGES2PKM
SCHEMBL31553928 0.83 KMT2A (0.38) KMT2ATRPV4PTGES2PKMTSHR
SCHEMBL16852853 0.83 KMT2A (0.38) KMT2ATRPV4PTGES2PKMTSHR
SCHEMBL23978197 0.81 CA2 (0.50) KMT2APTGES2CA12CA1CA2
SCHEMBL29545876 0.79 KMT2A (0.49) KMT2AEPHX2PTGES2PKMTSHR
SCHEMBL2369020 0.79 KMT2A (0.49) KMT2AEPHX2PTGES2PKMTSHR
SCHEMBL29899701 0.78 AKR1B1 (0.46) TRPV4PKMAKR1B1CCR2
SCHEMBL113810 0.78 AKR1B1 (0.46) TRPV4PKMAKR1B1CCR2
SCHEMBL31470482 0.78 HSP90AA1 (0.43) TRPV4EPHX2AKR1B1TSHRHTT
SCHEMBL1814581 0.78 HSP90AA1 (0.43) TRPV4EPHX2AKR1B1TSHRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 148 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104678028-A Pretreatment and detection method for biogen amine neurotransmitter and detection kit INST PHARM & TOXICOLOGY AMMS 2015-06-03 CN claimed
US-12565497-B2 Sulfone derivatives HOFFMANN-LA ROCHE INC. (US) 2026-03-03 US disclosed
US-20250282781-A1 APOL1 INHIBITORS AND METHODS OF USE HERCULES CAPITAL, INC., AS AGENT 2025-09-11 US disclosed
US-12344610-B2 APOL1 inhibitors and methods of use MAZE THERAPEUTICS, INC. (US) 2025-07-01 US disclosed
US-20250026721-A1 COMPOUNDS AND METHODS FOR MODULATING RAS-PI3K VIVIDION THERAPEUTICS, INC. 2025-01-23 US disclosed
WO-2024249254-A2 METHODS OF USING APOL1 INHIBITORS MAZE THERAPEUTICS, INC. (US) 2024-12-05 WO disclosed
US-20240400565-A1 APOL1 INHIBITORS AND METHODS OF USE HERCULES CAPITAL, INC., AS AGENT 2024-12-05 US disclosed
EP-4465982-A2 APOL1 INHIBITORS AND METHODS OF USE Maze Therapeutics, Inc. (US) 2024-11-27 EP disclosed
US-11976067-B2 APOL1 inhibitors and methods of use MAZE THERAPEUTICS, INC. (US) 2024-05-07 US disclosed
CN-117720498-A Synthesis of novel coumarin derivative containing sulfonamide fragments and preparation method and application of composition of novel coumarin derivative 贵州工业职业技术学院 2024-03-19 CN disclosed
EP-1797065-A2 ACYCLIC 1,3-DIAMINES AND USES THEREFOR SMITHKLINE BEECHAM CORPORATION (US) 2007-06-20 EP disclosed
WO-2006105475-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-05 WO disclosed
WO-2006029210-A2 ACYCLIC 1,3-DIAMINES AND USES THEREFOR SMITHKLINE BEECHAM CORPORATION (US) 2006-03-16 WO disclosed
US-20060052396-A1 Arylamines for the treatment of conditions associated with gsk-3 ASTRAZENECA (SE) 2006-03-09 US disclosed
EP-1549613-A1 SULFONAMIDES HAVING ANTIANGIOGENIC AND ANTICANCER ACTIVITY Abbott Laboratories (US) 2005-07-06 EP disclosed
US-20040167128-A1 Sulfonamides having antiangiogenic and anticancer activity ABBVIE INC. 2004-08-26 US disclosed
US-20040157836-A1 Sulfonamides having antiangiogenic and anticancer activity ABBOTT LABORATORIES 2004-08-12 US disclosed
EP-1414801-A1 ARYLAMINES FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH GSK-3 AstraZeneca AB (SE) 2004-05-06 EP disclosed
WO-2004033419-A1 SULFONAMIDES HAVING ANTIANGIOGENIC AND ANTICANCER ACTIVITY ABBOTT LABORATORIES (US) 2004-04-22 WO disclosed
WO-2003004472-A1 ARYLAMINES FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH GSK-3 ASTRAZENECA AB (SE) 2003-01-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250026721-A1 COMPOUNDS AND METHODS FOR MODULATING RAS-PI3K KRAS, HRAS, NRAS KMT2A 2722/4885TRPV4 4643/4885EPHX2 2121/4885
US-20040167128-A1 Sulfonamides having antiangiogenic and anticancer activity METAP2, METAP1, DNPEP KMT2A 647/4885TRPV4 3852/4885EPHX2 971/4885
US-12344610-B2 APOL1 inhibitors and methods of use APOL1, APOB, PON1 KMT2A 4701/4885TRPV4 4647/4885EPHX2 2968/4885
US-20040157836-A1 Sulfonamides having antiangiogenic and anticancer activity METAP2, METAP1, DNPEP KMT2A 647/4885TRPV4 3852/4885EPHX2 971/4885
US-11976067-B2 APOL1 inhibitors and methods of use APOL1, APOB, LDLR KMT2A 4715/4885TRPV4 4637/4885EPHX2 2977/4885
US-20250282781-A1 APOL1 INHIBITORS AND METHODS OF USE APOL1, APOB, PON1 KMT2A 4701/4885TRPV4 4647/4885EPHX2 2968/4885
US-20240400565-A1 APOL1 INHIBITORS AND METHODS OF USE APOL1, APOB, PON1 KMT2A 4701/4885TRPV4 4647/4885EPHX2 2968/4885
US-20060052396-A1 Arylamines for the treatment of conditions associated with gsk-3 GSK3A, GSK3B, PYGL KMT2A 686/4885TRPV4 3939/4885EPHX2 2850/4885
US-12565497-B2 Sulfone derivatives CXCR1, CCR1, SULT1E1 KMT2A 4321/4885TRPV4 2973/4885EPHX2 1721/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.