SCHEMBL4350090

SCHEMBL4350090

Oc1c(F)cc(Br)cc1NC(=S)NCCc1ccccc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.73
ALOX12 P18054 5/20 0.73
MEN1 O00255 4/20 0.73
KMT2A Q03164 4/20 0.73
MAPT P10636 4/20 0.73
CYP1A2 P05177 3/20 0.73
CYP2D6 P10635 3/20 0.73
CYP2C9 P11712 3/20 0.73
CYP2C19 P33261 3/20 0.73
CYP3A4 P08684 2/20 0.73
RAB9A P51151 6/20 0.64
NPC1 O15118 5/20 0.64
ALDH1A1 P00352 8/20 0.62
LMNA P02545 5/20 0.62
HTT P42858 1/20 0.62
HPGD P15428 2/20 0.60
POLB P06746 1/20 0.60
MAOA P21397 1/20 0.52
MAOB P27338 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4342066 0.87 ALOX12 (0.55) SMN1; SMN2ALOX12MEN1KMT2AMAPT
SCHEMBL4345936 0.85 MEN1 (0.53) SMN1; SMN2ALOX12MEN1KMT2AMAPT
SCHEMBL4355894 0.82 NPC1 (0.79) SMN1; SMN2ALOX12MEN1KMT2AMAPT
SCHEMBL4349029 0.80 RAB9A (0.68) SMN1; SMN2ALOX12MEN1KMT2AMAPT
SCHEMBL4348536 0.79 LMNA (0.69) SMN1; SMN2ALOX12MEN1KMT2AMAPT
SCHEMBL27761072 0.78 SMN1; SMN2 (0.57) SMN1; SMN2ALOX12MEN1KMT2AMAPT
SCHEMBL4346353 0.78 ALDH1A1 (0.80) SMN1; SMN2ALOX12MEN1KMT2AMAPT
SCHEMBL4349397 0.77 SMN1; SMN2 (0.52) SMN1; SMN2ALOX12MEN1KMT2AMAPT
SCHEMBL4345595 0.76 MEN1 (0.46) SMN1; SMN2ALOX12MEN1KMT2AMAPT
SCHEMBL4350009 0.75 RAB9A (0.68) SMN1; SMN2ALOX12MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110065760-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES AND USE THEREOF JERINI AG (DE) 2011-03-17 US claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
US-20070054904-A1 Phenol derivatives and their use as rotamase inhibitors JERINI AG (DE) 2007-03-08 US claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110065760-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES AND USE THEREOF NR1I3, NR1D1, NR1D2 SMN1; SMN2 1791/4885ALOX12 1546/4885MEN1 2168/4885
US-20070054904-A1 Phenol derivatives and their use as rotamase inhibitors NR1I3, NR1D1, NR1D2 SMN1; SMN2 3250/4885ALOX12 1994/4885MEN1 3901/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.