SCHEMBL4350353

SCHEMBL4350353

Cc1cccc2[nH]c(C3CN(C)CC[N]3)nc12

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.45
PARP1 P09874 5/20 0.43
PDE10A Q9Y233 2/20 0.43
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
HCRTR1 O43613 4/20 0.38
HCRTR2 O43614 4/20 0.38
MGAM O43451 5/20 0.38
GAA P10253 5/20 0.38
SI P14410 5/20 0.38
MGAM2 Q2M2H8 5/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4358956 0.86 PARP1 (0.45) PARP1GAA
SCHEMBL4344619 0.86 PARP1 (0.42) PARP1HCRTR1HCRTR2
SCHEMBL4350617 0.85 HCRTR1 (0.38) HRH4PARP1HCRTR1HCRTR2
SCHEMBL4098540 0.81 PARP1 (0.41) PARP1PTGS1PTGS2
SCHEMBL4097945 0.80 HRH4 (0.47) HRH4PARP1
SCHEMBL2201563 0.77 MGAM (0.40) PDE10APTGS1PTGS2HCRTR1HCRTR2
SCHEMBL4353639 0.76 KDM4E (0.40) HCRTR1HCRTR2GAA
SCHEMBL4348250 0.74 LMNA (0.39) HRH4PDE10A
SCHEMBL4358835 0.73 SSTR5 (0.36) HRH4PARP1
SCHEMBL4103942 0.72 KCNH2 (0.40) HRH4HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504426-B2 Heterocyclic compounds JANSSEN PHARMACEUTICA N.V. (BE) 2009-03-17 US disclosed