SCHEMBL4344619

SCHEMBL4344619

CN1CC[N]C(c2nc3c(Cl)cccc3[nH]2)C1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.42
PSMB8 P28062 1/20 0.39
HCRTR1 O43613 10/20 0.38
HCRTR2 O43614 10/20 0.38
PARP2 Q9UGN5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4350353 0.86 HRH4 (0.45) PARP1HCRTR1HCRTR2
SCHEMBL4358956 0.85 PARP1 (0.45) PARP1PARP2
SCHEMBL4098540 0.80 PARP1 (0.41) PARP1PARP2
SCHEMBL4350617 0.79 HCRTR1 (0.38) PARP1HCRTR1HCRTR2
SCHEMBL4356646 0.77 HRH4 (0.45) HCRTR1HCRTR2
SCHEMBL4097945 0.77 HRH4 (0.47) PARP1
SCHEMBL4356635 0.75 HRH4 (0.47)
SCHEMBL4103942 0.74 KCNH2 (0.40) HCRTR1HCRTR2
SCHEMBL4358835 0.72 SSTR5 (0.36) PARP1
SCHEMBL4348250 0.71 LMNA (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504426-B2 Heterocyclic compounds JANSSEN PHARMACEUTICA N.V. (BE) 2009-03-17 US disclosed