SCHEMBL4351360

SCHEMBL4351360

CC(C)(C)OC(=O)N1CCC(C2OCc3cc(-c4ccc(C(=O)N5CCN(CCO)CC5)cn4)ccc3O2)CC1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 14/20 0.42
HRH3 Q9Y5N1 2/20 0.39
CRBN Q96SW2 1/20 0.38
DYRK2 Q92630 1/20 0.38
STAT3 P40763 1/20 0.38
HDAC4 P56524 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4354311 0.93 GPR119 (0.44) GPR119CRBNDYRK2STAT3HDAC4
SCHEMBL4347903 0.89 GPR119 (0.44) GPR119HRH3
SCHEMBL4525904 0.89 HRH3 (0.40) GPR119HRH3STAT3
SCHEMBL4352666 0.87 GPR119 (0.49) GPR119DYRK2
SCHEMBL4536512 0.86 GPR119 (0.47) GPR119
SCHEMBL4355704 0.84 RAB9A (0.46) HRH3STAT3
SCHEMBL13586034 0.83 ABL1 (0.46) GPR119CRBNHDAC4
SCHEMBL4352054 0.82 GPR119 (0.46) GPR119
SCHEMBL4536116 0.81 STAT3 (0.43) HRH3STAT3
SCHEMBL13586046 0.80 GPR119 (0.57) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150144-A1 NEW GPR119MODULATORS INOVACIA AB (SE) 2009-12-17 WO disclosed
WO-2009150144-A1 NEW GPR119MODULATORS INOVACIA AB (SE) 2009-12-17 WO disclosed