SCHEMBL4358291

SCHEMBL4358291

COC(=O)c1sccc1S(N)(=O)=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CA5A P35218 1/20 0.51
CA9 Q16790 1/20 0.51
EDNRA P25101 3/20 0.51
MAPT P10636 4/20 0.49
TP53 P04637 1/20 0.49
KMT2A Q03164 2/20 0.49
LMNA P02545 4/20 0.48
POLB P06746 2/20 0.48
THRB P10828 1/20 0.48
HPGD P15428 1/20 0.48
TSHR P16473 1/20 0.48
NPC1 O15118 1/20 0.47
MEN1 O00255 1/20 0.46
CYP1A2 P05177 1/20 0.46
KCNH2 Q12809 1/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
PPARG P37231 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18920867 0.87 CA1 (0.43) CA1CA2CA5ACA9EDNRA
SCHEMBL23569071 0.87 EDNRA (0.49) EDNRAMAPTTP53KMT2ALMNA
SCHEMBL23569216 0.85 EDNRA (0.48) EDNRAMAPTTP53KMT2ALMNA
SCHEMBL11471141 0.84 EDNRA (0.52) EDNRAMAPTTP53KMT2ALMNA
SCHEMBL12319426 0.84 EDNRA (0.52) EDNRAMAPTTP53KMT2ALMNA
SCHEMBL388034 0.83 MAPT (0.55) EDNRAMAPTTP53KMT2ALMNA
SCHEMBL31607236 0.83 EDNRA (0.51) EDNRAMAPTTP53KMT2ALMNA
SCHEMBL8973588 0.82 PKM (0.45) CA1CA2CA9MAPTKMT2A
SCHEMBL11469582 0.81 EDNRA (0.56) EDNRAMAPTTP53KMT2ALMNA
SCHEMBL11117907 0.81 EDNRA (0.53) EDNRAMAPTTP53KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 86 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170043196-A1 Fire Extinguishing Composition Comprising Heterocyclic Compounds XI'AN J&R FIRE FIGHTING EQUIPMENT CO., LTD. (CN) 2017-02-16 US claimed
EP-3095485-A1 FIRE EXTINGUISHING COMPOSITION COMPRISING HETEROCYCLIC COMPOUNDS Xi'an J&R Fire Fighting Equipment Co., Ltd. (CN) 2016-11-23 EP claimed
CN-102020667-B Method for synthesizing 6-chloro-4-hydroxyl-2-methyl-2H-thieno(2.3.e)-1.2thiazide-1.1-dioxide-3-methyl formate LIU YULIN 2013-02-27 CN claimed
EP-3986879-B1 FUSED 1,2-THIAZOLES AND 1,2-THIAZINES WHICH ACT AS NLRP3 MODULATORS AC IMMUNE SA (CH) 2024-10-02 EP disclosed
EP-4276092-A1 COMPOUND LIBRARY CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2023-11-15 EP disclosed
CN-116783160-A Libraries of compounds 中外制药株式会社 2023-09-19 CN disclosed
US-20220378801-A1 NOVEL COMPOUNDS AC IMMUNE SA (CH) 2022-12-01 US disclosed
EP-3986879-A1 FUSED 1,2 THIAZOLES AND 1,2 THIAZINES WHICH ACT AS NL3P3 MODULATORS AC Immune SA (CH) 2022-04-27 EP disclosed
CN-114008030-A Fused 1, 2-thiazoles and 1, 2-thiazines as NLRP3 modulators AC免疫有限公司 2022-02-01 CN disclosed
WO-2021123237-A1 2-AMINO-N-(AMINO-OXO-ARYL-LAMBDA6-SULFANYLIDENE)ACETAMIDE COMPOUNDS AND THEIR THERAPEUTIC USE Oxford Drug Design Limited (GB) 2021-06-24 WO disclosed
WO-2020254697-A1 FUSED 1,2 THIAZOLES AND 1,2 THIAZINES WHICH ACT AS NL3P3 MODULATORS AC IMMUNE SA (CH) 2020-12-24 WO disclosed
US-4877440-A Thiophenesulfonamide herbicides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1989-10-31 US disclosed
US-4743290-A Thiophenesulfonamide herbicides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1988-05-10 US disclosed
US-4701535-A CHEMICAL INTERMEDIATES FOR HERBICIDES, PLANT GROWTH REGULATOR E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-10-20 US disclosed
EP-0207609-A1 Herbicidal thiophenesulfonamides E.I. DU PONT DE NEMOURS AND COMPANY (US) 1987-01-07 EP disclosed
US-4599103-A PRE-AND POSTEMERGENCE HERBICIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 1986-07-08 US disclosed
EP-0030142-B1 HERBICIDAL UREAS, PREPARATION, COMPOSITIONS AND USE THEREOF E.I. DU PONT DE NEMOURS AND COMPANY (US) 1984-12-05 EP disclosed
US-4481029-A HERBICIDES, PLANT GROWTH REGULATORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1984-11-06 US disclosed
EP-0030142-A2 Herbicidal ureas, preparation, compositions and use thereof E.I. DU PONT DE NEMOURS AND COMPANY (US) 1981-06-10 EP disclosed
US-4028373-A ARTIFICIAL SWEETNERS BASF AKTIENGESELLSCHAFT (DT) 1977-06-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220378801-A1 NOVEL COMPOUNDS NLRP3, IL1B, IL18 CA1 4311/4885CA2 4210/4885CA5A 2377/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.