SCHEMBL4358362

SCHEMBL4358362

CCCNc1nc(N)nc2ccc(-c3ccc(OC)c(OC)c3)cc12

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
APP P05067 7/20 0.57
BCHE P06276 3/20 0.49
ACHE P22303 3/20 0.49
DHFR P00374 3/20 0.47
TLR7 Q9NYK1 4/20 0.45
TLR8 Q9NR97 2/20 0.45
CLK4 Q9HAZ1 1/20 0.43
PDE5A O76074 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
KCNH2 Q12809 1/20 0.41
FYN P06241 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4362251 0.93 APP (0.55) APPDHFRTLR7TLR8ALDH1A1
SCHEMBL4367762 0.87 APP (0.54) APPBCHEACHEDHFRTLR7
SCHEMBL4074235 0.84 NOS1 (0.48) APPTLR7FYN
SCHEMBL4357089 0.84 APP (0.50) APPDHFRCLK4KDM4E
SCHEMBL4358329 0.81 APP (0.59) APPTLR7TLR8PDE5AKCNH2
SCHEMBL4355328 0.81 APP (0.59) APPTLR7TLR8PDE5A
SCHEMBL4354805 0.81 CLK4 (0.64) APPCLK4ALDH1A1
SCHEMBL4358891 0.80 ACHE (0.62) APPBCHEACHECLK4PDE5A
SCHEMBL4351984 0.79 NSD2 (0.56) APPBCHEACHEDHFRCLK4
SCHEMBL4362768 0.78 DHFR (0.69) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 56 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12049461-B2 4,6-di- and 2,4,6-trisubstituted quinazoline derivatives useful for treating viral infections GILEAD SCIENCES, INC. (US) 2024-07-30 US claimed
US-20210276988-A1 4,6-DI- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. 2021-09-09 US claimed
US-10882851-B2 4,6-di- and 2,4,6-trisubstituted quinazoline derivatives useful for treating viral infections GILEAD SCIENCES, INC. (US) 2021-01-05 US claimed
US-20160257673-A1 4,6-DI- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. 2016-09-08 US claimed
US-9259426-B2 4,6-di- and 2,4,6-trisubstituted quinazoline derivatives useful for treating viral infections GILEAD SCIENCES, INC. (US) 2016-02-16 US claimed
US-20090285782-A1 4,6-DI- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2009-11-19 US claimed
US-12049461-B2 4,6-di- and 2,4,6-trisubstituted quinazoline derivatives useful for treating viral infections GILEAD SCIENCES, INC. (US) 2024-07-30 US disclosed
US-20240134300-A1 TONER CANON KABUSHIKI KAISHA (JP) 2024-04-25 US disclosed
CN-111630456-B White toner 佳能株式会社 2024-04-16 CN disclosed
CN-117850181-A Toner and method for producing the same 佳能株式会社 2024-04-09 CN disclosed
US-20240067593-A1 PRODUCTION OF AROMATIC ACIDS AND PHENOLICS NEDERLANDSE ORGANISATIE VOOR TOEGEPAST-NATUURWETENSCHAPPELIJK ONDERZOEK TNO (NL) 2024-02-29 US disclosed
EP-4048652-B1 PRODUCTION OF AROMATIC ACIDS AND PHENOLICS TNO (NL) 2023-10-04 EP disclosed
US-20230088424-A1 TONER PROCESSING APPARATUS AND METHOD FOR PRODUCING TONER CANON KABUSHIKI KAISHA (JP) 2023-03-23 US disclosed
US-6232277-B1 ETHYLENE POLYMER; CONDENSATION PRODUCT OF ALDEHYDE OR KETONE WITH HYDROXY-, ALKOXY-, MERCAPTO-AND/OR ALKYLTHIO-SUBSTITUTED ALKYLARYL COMPOUND; AND POLAR NITROGEN COMPOUND; COLD FLOW, FILTERABILITY EXXON CHEMICAL PATENTS INC 2001-05-15 US disclosed
EP-1088013-A1 ADDITIVES AND OIL COMPOSITIONS Infineum USA L.P. (US) 2001-04-04 EP disclosed
EP-1088045-A1 ADDITIVES AND OIL COMPOSITIONS Infineum USA L.P. (US) 2001-04-04 EP disclosed
WO-1999061562-A1 ADDITIVES AND OIL COMPOSITIONS INFINEUM USA L.P. (US) 1999-12-02 WO disclosed
WO-1999061498-A1 ADDITIVES AND OIL COMPOSITIONS INFINEUM USA L.P. (US) 1999-12-02 WO disclosed
US-4606947-A HYDROXYL CONTAINING POLYESTER AND POLYISOCYANATE BLOCKED WITH ACETOACETIC ACID ALKYL ESTER HERBERTS GMBH (DE) 1986-08-19 US disclosed
US-4367295-A POLYURETHANES BAYER AKTIENGESELLSCHAFT (DE) 1983-01-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12049461-B2 4,6-di- and 2,4,6-trisubstituted quinazoline derivatives useful for treating viral infections NR3C1, NR3C2, NR4A1 APP 4361/4885BCHE 4599/4885ACHE 4515/4885
US-20210276988-A1 4,6-DI- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR TREATING VIRAL INFECTIONS NR3C1, NR3C2, NR4A1 APP 4361/4885BCHE 4599/4885ACHE 4515/4885
US-20240067593-A1 PRODUCTION OF AROMATIC ACIDS AND PHENOLICS DDC, PAH, FDPS APP 895/4885BCHE 4019/4885ACHE 1252/4885
US-20090285782-A1 4,6-DI- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR TREATING VIRAL INFECTIONS NR3C1, NR5A2, NR4A1 APP 4235/4885BCHE 4565/4885ACHE 4468/4885
US-10882851-B2 4,6-di- and 2,4,6-trisubstituted quinazoline derivatives useful for treating viral infections NR3C1, NR3C2, NR5A2 APP 4318/4885BCHE 4694/4885ACHE 4535/4885
US-20160257673-A1 4,6-DI- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR TREATING VIRAL INFECTIONS NR3C1, NR3C2, NR5A2 APP 4318/4885BCHE 4694/4885ACHE 4535/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.