SCHEMBL4358469

SCHEMBL4358469

CCN1CC[N]C(c2nc3cc(F)c(F)cc3[nH]2)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.38
HRH4 Q9H3N8 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
MPO P05164 1/20 0.37
OPRL1 P41146 5/20 0.36
KCNH2 Q12809 2/20 0.36
ALDH1A1 P00352 2/20 0.32
PRCP P42785 1/20 0.32
KDM4E B2RXH2 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
CYP2C19 P33261 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
CAMK2D Q13557 1/20 0.31
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4354354 0.84 HRH4 (0.44) PDE10AHRH4HRH3MPOOPRL1
SCHEMBL4109197 0.71 TXN (0.36) PDE10AHRH4HRH3OPRL1KCNH2
SCHEMBL4353639 0.69 KDM4E (0.40) ALDH1A1KDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL4350354 0.69 MPO (0.38) PDE10AHRH4HRH3MPOOPRL1
SCHEMBL4356646 0.68 HRH4 (0.45) HRH4PRCPKDM4ECYP1A2CYP3A4
SCHEMBL4103942 0.66 KCNH2 (0.40) HRH4KCNH2HCRTR1HCRTR2
SCHEMBL4348250 0.65 LMNA (0.39) PDE10AHRH4ALDH1A1KDM4ECYP1A2
SCHEMBL4352227 0.64 HRH4 (0.35) HRH4HRH3ALDH1A1HCRTR1HCRTR2
SCHEMBL4356635 0.64 HRH4 (0.47) HRH4HRH3ALDH1A1
SCHEMBL604024 0.64 HRH4 (0.60) HRH4HRH3OPRL1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504426-B2 Heterocyclic compounds JANSSEN PHARMACEUTICA N.V. (BE) 2009-03-17 US disclosed