SCHEMBL4356646

SCHEMBL4356646

CN1CC[N]C(c2nc3cc(Cl)c(Cl)cc3[nH]2)C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.45
CACNA1G O43497 1/20 0.41
CACNA1H O95180 1/20 0.41
PRCP P42785 11/20 0.40
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
KDM4E B2RXH2 1/20 0.38
GMNN O75496 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
BLM P54132 1/20 0.38
PMP22 Q01453 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.38
NFKB1 P19838 1/20 0.38
STAT6 P42226 1/20 0.38
HIF1A Q16665 1/20 0.38
AR P10275 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4103942 0.91 KCNH2 (0.40) HRH4HCRTR1HCRTR2
SCHEMBL4353639 0.85 KDM4E (0.40) GAAHTTKDM4ELMNAMAPT
SCHEMBL4356635 0.85 HRH4 (0.47) HRH4GAAHTTLMNAMAPT
SCHEMBL4354354 0.84 HRH4 (0.44) HRH4PRCPKDM4ECYP1A2CYP3A4
SCHEMBL4109197 0.83 TXN (0.36) HRH4CACNA1GCACNA1HPRCPHCRTR1
SCHEMBL4348250 0.81 LMNA (0.39) HRH4HTTKDM4ELMNAMAPT
SCHEMBL4352227 0.80 HRH4 (0.35) HRH4HTTLMNAHCRTR1HCRTR2
SCHEMBL4350354 0.80 MPO (0.38) HRH4KDM4EHCRTR1HCRTR2
SCHEMBL4355101 0.78 ALDH1A1 (0.38) HRH4GAAMAPTSMN1; SMN2CYP1A2
SCHEMBL4344619 0.77 PARP1 (0.42) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504426-B2 Heterocyclic compounds JANSSEN PHARMACEUTICA N.V. (BE) 2009-03-17 US disclosed