SCHEMBL4359570

SCHEMBL4359570

CCOc1ccc(-n2[nH]c(=O)c3cc(NS(=O)(=O)c4cccc(C(F)(F)F)c4)ccc32)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 2/20 0.48
AR P10275 2/20 0.48
PGR P06401 1/20 0.48
ESR2 Q92731 1/20 0.48
HIF1A Q16665 1/20 0.47
HSD17B2 P37059 1/20 0.45
POLB P06746 1/20 0.44
LMNA P02545 3/20 0.43
PKM P14618 2/20 0.43
HTT P42858 1/20 0.43
MAPT P10636 2/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
HTR6 P50406 2/20 0.42
BRAF P15056 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ALOX15 P16050 1/20 0.42
TOP2A P11388 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4362689 0.81 POLB (0.48) POLBLMNAPKMHTTMAPT
SCHEMBL3908386 0.79 HSD17B2 (0.50) NR3C1ARPGRESR2HIF1A
SCHEMBL4370085 0.78 ALOX15 (0.42) HIF1APOLBLMNAPKMHTT
SCHEMBL3909496 0.77 HSD17B2 (0.49) NR3C1ARPGRESR2HIF1A
SCHEMBL4363789 0.76 ALDH1A1 (0.53) HSD17B2POLBLMNAHTTMAPT
SCHEMBL1807440 0.75 NR3C1 (0.51) NR3C1ARPGRESR2HIF1A
SCHEMBL3917148 0.73 NR3C1 (0.48) NR3C1ARPGRESR2HIF1A
SCHEMBL27180227 0.72 POLB (0.60) NR3C1ARPGRESR2POLB
SCHEMBL27678794 0.72 HDAC1 (0.50) NR3C1ARPGRESR2HIF1A
SCHEMBL1821354 0.71 BRD4 (0.59) PGRHSD17B2MAPTHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797042-B1 INDOZOLONE DERIVATIVES AS 11B-HSD1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-01-07 EP claimed