SCHEMBL4373471

SCHEMBL4373471

O=C(O)N1CCC(CNc2cnc(-c3ccc(C(=O)N4CCC(O)C4)cc3)cn2)CC1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ATR Q13535 4/20 0.50
TPH1 P17752 2/20 0.48
TBK1 Q9UHD2 1/20 0.44
VNN1 O95497 3/20 0.43
HDAC4 P56524 1/20 0.42
PIM1 P11309 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
GRIN2B Q13224 1/20 0.39
GABRA5 P31644 1/20 0.39
CYP11B2 P19099 1/20 0.39
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
HTR2B P41595 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4371541 0.96 TPH1 (0.48) ATRTPH1TBK1VNN1HDAC4
SCHEMBL13690341 0.86 GPR119 (0.49) ATRTPH1TBK1
SCHEMBL4050033 0.86 TPH1 (0.53) ATRTPH1PIM1CYP3A4CYP2D6
SCHEMBL4056100 0.85 TPH1 (0.44) ATRTPH1TBK1VNN1PIM1
SCHEMBL4234932 0.84 TPH1 (0.49) ATRTPH1PIM1CYP3A4CYP2D6
SCHEMBL13690750 0.83 GPR119 (0.49) TPH1
SCHEMBL4376173 0.82 ATR (0.48) ATRVNN1HDAC4GABRA5ALOX5AP
SCHEMBL4057216 0.82 IKBKB (0.48) ATRTPH1VNN1
SCHEMBL4370900 0.82 IKBKB (0.48) ATRTPH1VNN1
SCHEMBL4379368 0.82 TPH1 (0.44) ATRTPH1PIM1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009106561-A1 PYRAZINE COMPOUNDS FOR TREATING GPR119 RELATED DISORDERS BIOVITRUM AB (PUBL) (SE) 2009-09-03 WO disclosed