SCHEMBL437482

SCHEMBL437482

Cc1ccc(Cl)c2c(N)c(Cl)cnc12

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.35
MAPT P10636 3/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
LMNA P02545 1/20 0.34
KDM4E B2RXH2 2/20 0.33
POLB P06746 2/20 0.33
CCR1 P32246 1/20 0.31
CCR5 P51681 1/20 0.31
CCR8 P51685 1/20 0.31
NOS3 P29474 1/20 0.31
NOS2 P35228 1/20 0.31
HAVCR2 Q8TDQ0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL436692 0.91 POLB (0.38) CYP3A4MAPTMEN1KMT2ALMNA
SCHEMBL436747 0.84 CYP3A4 (0.32) CYP3A4MAPTMEN1KMT2ALMNA
SCHEMBL437555 0.84 HAVCR2 (0.38) CYP3A4HAVCR2
SCHEMBL442158 0.79 HAVCR2 (0.54) MAPTMEN1KMT2ALMNAKDM4E
SCHEMBL439519 0.77 DYRK1A (0.39) MAPTMEN1KMT2AKDM4EPOLB
SCHEMBL440196 0.74 NPC1 (0.52) MAPTMEN1KMT2ALMNAKDM4E
SCHEMBL442075 0.73 HAVCR2 (0.46) MAPTMEN1KMT2ALMNAKDM4E
SCHEMBL437847 0.73 CCR1 (0.42) CYP3A4MAPTKMT2ALMNAKDM4E
SCHEMBL15146338 0.71 CCR1 (0.45) CYP3A4MAPTMEN1KMT2ALMNA
SCHEMBL436942 0.70 HAVCR2 (0.41) MAPTMEN1KMT2ACCR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed